REGIOSELECTIVE ALKYLATION OF THE EXOCYCLIC NITROGEN OF HETEROCYCLIC AMIDINES VIA THE MITSUNOBU REACTION

被引：16

作者：

ABARGHAZ, M

KERBAL, A

BOURGUIGNON, JJ

机构：

[1] CTR NEUROCHIM,CNRS,PHARMACOCHIM MOLEC LAB,F-67084 STRASBOURG,FRANCE

[2] FAC SCI DHAR EL MEHRAZ,CHIM ORGAN LAB,ATLAS FES,MOROCCO

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 36期

关键词：

D O I：

10.1016/0040-4039(95)01304-Z

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Regioselective alkylation of heterocyclic amidines by means of Mitsunobu reaction leads to L-aminoacid derivatives.

引用

页码：6463 / 6466

页数：4

共 18 条

[1] METHYLATION OF PROTOMERIC AMBIDENT NUCLEOPHILES WITH METHYL FLUOROSULFONATE - REGIOSPECIFIC REACTION [J].

BEAK, P ;

LEE, JK ;

MCKINNIE, BG .

JOURNAL OF ORGANIC CHEMISTRY, 1978, 43 (07) :1367-1372

[2] EXPERIMENTAL-EVIDENCE FOR GEOMETRICAL VARIATIONS IN TRANSITION-STATE OF SN2 REACTION [J].

BERG, U ;

GALLO, R ;

METZGER, J ;

CHANON, M .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1976, 98 (05) :1260-1262

[3] ALPHA-ALKYLAMINOPYRIDINES AND 1,5-DI-(ALKYL-ALPHA-PYRIDYLAMINO)-PENTANES [J].

BLICKE, FF ;

TSAO, MU .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1946, 68 (05) :905-906

[4] CHIRAL AZOLE DERIVATIVES .2. SYNTHESIS OF ENANTIOMERICALLY PURE 1-ALKYLIMIDAZOLES [J].

CORELLI, F ;

SUMMA, V ;

BROGI, A ;

MONTEAGUDO, E ;

BOTTA, M .

JOURNAL OF ORGANIC CHEMISTRY, 1995, 60 (07) :2008-2015

[5] AN ABINITIO STUDY OF PROTONATION AND ALKYLATION OF AMINOPYRIDINE [J].

FOSSEY, J ;

LOUPY, A ;

STRZELECKA, H .

TETRAHEDRON, 1981, 37 (10) :1935-1941

[6] UBER DIE ALKYLIERUNG EINIGER AMINOHETEROCYCLEN UND DIE UMLAGERUNG HETEROCYCLISCHER IMINE IN AMINE [J].

GOERDELER, J ;

ROTH, W .

CHEMISCHE BERICHTE-RECUEIL, 1963, 96 (02) :534-&

[7] SYNTHETIC ROUTES TO NUCLEOSIDE ANALOGS OF N-SUBSTITUTED 1,3-THIAZOLIDINES [J].

IWAKAWA, M ;

PINTO, BM ;

SZAREK, WA .

CANADIAN JOURNAL OF CHEMISTRY-REVUE CANADIENNE DE CHIMIE, 1978, 56 (03) :326-335

[8]

MAGHIOROS G, 1983, NOUV J CHIM, V7, P667

[9]

MAGIDSON O, BER, V59, P1209

[10] STEREOSPECIFIC AND STEREOSELECTIVE REACTIONS .1. PREPARATION OF AMINES FROM ALCOHOLS [J].

MITSUNOB.O ;

WADA, M ;

SANO, T .

JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1972, 94 (02) :679-&

← 1 2 →