SYNTHESIS AND ANTIMICROBIOLOGICAL ACTIVITY OF N-ARYL-SUBSTITUTED 2-METHYL-3-CARBETHOXY-5-PYRROLINONE DERIVATIVES

被引：4

作者：

LOVREN, F ^{[1
]}

GAON, ID ^{[1
]}

BOBAREVIC, B ^{[1
]}

机构：

[1] FAC MED SARAJEVO, DEPT MED CHEM, YU-71000 SARAJEVO, YUGOSLAVIA

来源：

ARCHIV DER PHARMAZIE | 1990年 / 323卷 / 11期

关键词：

D O I：

10.1002/ardp.19903231104

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

We describe the synthesis of N‐aryl‐2‐methyl‐3‐carbethoxy‐5‐pyrrolinones benzylidene derivatives, their condensation with azomethines and substitution with aniline. The compounds have been tested for antimicrobial and fungicide activity: they have better fungicidal than bactericidal activity. Copyright © 1990 WILEY‐VCH Verlag GmbH & Co. KGaA, Weinheim

引用

页码：901 / 904

页数：4

共 8 条

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[3]

FILACCHIONI G, 1983, FARMACO-ED SCI, V38, P619

[4]

GALDINO SL, 1986, FARMACO, V41, P59

[5]

GAON ID, 1985, FARM VEST, V36, P221

[6]

GAON ID, 1986, FARM VESTN, V37, P241

[7]

LOVREN F, 1988, ACTA PHARM JUGOSL, V38, P123

[8]

THIAULT GA, 1984, FARMACO-ED SCI, V39, P765

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