A NOVEL ASYMMETRIC-SYNTHESIS OF S-(+)-2-AMINO-4-PHOSPHONOBUTANOIC ACID

被引：13

作者：

JIAO, XY ^{[1
]}

CHEN, WY ^{[1
]}

HU, BF ^{[1
]}

机构：

[1] BEIJING AGR UNIV,INST APPL CHEM,BEIJING 100094,PEOPLES R CHINA

来源：

SYNTHETIC COMMUNICATIONS | 1992年 / 22卷 / 08期

关键词：

D O I：

10.1080/00397919208021103

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A novel asymmetric synthetic route to S(+)-2-amino-4-phosphonobutanoic acid through the cyclic condensation of ethyl-4-diethoxyphosphonyl-2-oxo-butanoate with L-erythro-(+)-1,2-diphenyl-2-hydroxyethylamine, followed by reduction and hydrolysis is described.

引用

页码：1179 / 1186

页数：8

共 11 条

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