SYNTHESIS OF CYCLIC-PEPTIDES VIA EFFICIENT NEW COUPLING REAGENTS

被引：56

作者：

EHRLICH, A ^{[1
]}

ROTHEMUND, S ^{[1
]}

BRUDEL, M ^{[1
]}

BEYERMANN, M ^{[1
]}

CARPINO, LA ^{[1
]}

BIENERT, M ^{[1
]}

机构：

[1] UNIV MASSACHUSETTS,DEPT CHEM,AMHERST,MA 01003

来源：

TETRAHEDRON LETTERS | 1993年 / 34卷 / 30期

关键词：

D O I：

10.1016/S0040-4039(00)74087-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The efficiency of various coupling reagents in promoting the cyclization of linear peptides has been compared. Newly developed reagents based on 1-hydroxy-7-azabenzotriazole were found to be highly effective and led to remarkably diminished racemization.

引用

页码：4781 / 4784

页数：4

共 19 条

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