SUPERIOR ANTIMALARIAL ACTIVITY OF PROGUANIL TO CYCLOGUANIL AFTER INVITRO BIOCONVERSION

被引:4
作者
RAMANAIAH, TV
机构
关键词
D O I
10.1016/0035-9203(88)90115-0
中图分类号
R1 [预防医学、卫生学];
学科分类号
1004 ; 120402 ;
摘要
引用
收藏
页码:358 / 359
页数:2
相关论文
共 7 条
[1]   METHODS FOR DETECTING CARCINOGENS AND MUTAGENS WITH SALMONELLA-MAMMALIAN-MICROSOME MUTAGENICITY TEST [J].
AMES, BN ;
MCCANN, J ;
YAMASAKI, E .
MUTATION RESEARCH, 1975, 31 (06) :347-363
[2]  
GAJANANA A, 1982, INDIAN J MED RES, V75, P802
[3]   A COMPARISON OF THE PYRIMETHAMINE AND CYCLOGUANIL SENSITIVITIES OF THE PRE-ERYTHROCYTIC AND ERYTHROCYTIC STAGES OF DRUG-SENSITIVE AND DRUG-RESISTANT STRAINS OF PLASMODIUM-YOELII [J].
HOWELLS, RE ;
GILLES, HM ;
BENT, NS .
ANNALS OF TROPICAL MEDICINE AND PARASITOLOGY, 1985, 79 (03) :247-251
[4]  
RAMANAIAH TV, 1985, CURR SCI INDIA, V54, P279
[5]   ANTIMALARIAL ACTIVITY AND METABOLISM OF BIGUANIDES .1. METABOLISM OF CHLORGUANIDE AND CHLORGUANIDE TRIAZINE IN RHESUS MONKEYS AND MAN [J].
SMITH, CC ;
MENNE, R ;
IHRIG, J .
AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE, 1961, 10 (05) :694-&
[6]  
THOMPSON PE, 1972, ANTIMALARIAL AGENTS, V12, P251
[7]   THE ACTIVITY OF PROGUANIL AND ITS METABOLITES, CYCLOGUANIL AND PARA-CHLOROPHENYLBIGUANIDE, AGAINST PLASMODIUM-FALCIPARUM INVITRO [J].
WATKINS, WM ;
SIXSMITH, DG ;
CHULAY, JD .
ANNALS OF TROPICAL MEDICINE AND PARASITOLOGY, 1984, 78 (03) :273-278