SYNTHESIS OF HYDROXAMIC ACIDS - PD/BASO4 AS A NEW CATALYST FOR THE DEPROTECTION OF O-BENZYL HYDROXAMATES

被引：58

作者：

NIKAM, SS

KORNBERG, BE

JOHNSON, DR

DOHERTY, AM

机构：

[1] Department of Chemistry, Parke-Davis Pharmaceutical Research Division, Warner-Lambert Company, Ann Arbor, MI 48105

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 02期

关键词：

D O I：

10.1016/0040-4039(94)02246-8

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Pd/BaSO4 was found to be an efficient catalyst in the deprotection of O-benzyl hydroxamates via hydrogenation to give the corresponding hydroxamic acids without further reduction to amides.

引用

页码：197 / 200

页数：4

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