PHENCYCLIDINE BLOCKS HISTAMINE H-3-RECEPTORS IN RAT-BRAIN

被引:25
作者
ARRANG, JM [1 ]
DEFONTAINE, N [1 ]
SCHWARTZ, JC [1 ]
机构
[1] CTR PAUL BROCA, NEUROBIOL & PHARMACOL UNITE, INSERM, U109, 2TER RUE ALESIA, F-75014 PARIS, FRANCE
关键词
D O I
10.1016/0014-2999(88)90467-0
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:31 / 35
页数:5
相关论文
共 30 条
[1]   THE BEHAVIORAL-EFFECTS OF PHENCYCLIDINES MAY BE DUE TO THEIR BLOCKADE OF POTASSIUM CHANNELS [J].
ALBUQUERQUE, EX ;
AGUAYO, LG ;
WARNICK, JE ;
WEINSTEIN, H ;
GLICK, SD ;
MAAYANI, S ;
ICKOWICZ, RK ;
BLAUSTEIN, MP .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (12) :7792-7796
[2]   AUTO-INHIBITION OF BRAIN HISTAMINE-RELEASE MEDIATED BY A NOVEL CLASS (H-3) OF HISTAMINE-RECEPTOR [J].
ARRANG, JM ;
GARBARG, M ;
SCHWARTZ, JC .
NATURE, 1983, 302 (5911) :832-837
[3]   AUTO-REGULATION OF HISTAMINE-RELEASE IN BRAIN BY PRESYNAPTIC H-3-RECEPTORS [J].
ARRANG, JM ;
GARBARG, M ;
SCHWARTZ, JC .
NEUROSCIENCE, 1985, 15 (02) :553-562
[4]   AUTOINHIBITION OF HISTAMINE SYNTHESIS MEDIATED BY PRESYNAPTIC H-3 RECEPTORS [J].
ARRANG, JM ;
GARBARG, M ;
SCHWARTZ, JC .
NEUROSCIENCE, 1987, 23 (01) :149-157
[5]   HIGHLY POTENT AND SELECTIVE LIGANDS FOR HISTAMINE RECEPTORS-H-3 [J].
ARRANG, JM ;
GARBARG, M ;
LANCELOT, JC ;
LECOMTE, JM ;
POLLARD, H ;
ROBBA, M ;
SCHUNACK, W ;
SCHWARTZ, JC .
NATURE, 1987, 327 (6118) :117-123
[6]   PHENCYCLIDINE-INDUCED RELEASE OF [H-3]DOPAMINE FROM CHOPPED STRIATAL TISSUE [J].
ARY, TE ;
KOMISKEY, HL .
NEUROPHARMACOLOGY, 1982, 21 (07) :639-645
[7]  
BALSTER RL, 1987, PSYCHOPHARMACOLOGY 3, P1573
[8]   PHENCYCLIDINE IN NANOMOLAR CONCENTRATIONS BINDS TO SYNAPTOSOMES AND BLOCKS CERTAIN POTASSIUM CHANNELS [J].
BLAUSTEIN, MP ;
ICKOWICZ, RK .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1983, 80 (12) :3855-3859
[9]   EFFECTS OF NALOXONE, METENKEPHALIN, AND MORPHINE ON PHENCYCLIDINE-INDUCED BEHAVIOR IN THE RAT [J].
CASTELLANI, S ;
GIANNINI, AJ ;
ADAMS, PM .
PSYCHOPHARMACOLOGY, 1982, 78 (01) :76-80
[10]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099