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Farnesyl transferase inhibitors: The successes and surprises of a new class of potential cancer chemotherapeutics
被引:63
作者
:
Buss, JE
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC,DEPT BIOORGAN CHEM,S SAN FRANCISCO,CA 94080
GENENTECH INC,DEPT BIOORGAN CHEM,S SAN FRANCISCO,CA 94080
Buss, JE
[
1
]
Marsters, JC
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC,DEPT BIOORGAN CHEM,S SAN FRANCISCO,CA 94080
GENENTECH INC,DEPT BIOORGAN CHEM,S SAN FRANCISCO,CA 94080
Marsters, JC
[
1
]
机构
:
[1]
GENENTECH INC,DEPT BIOORGAN CHEM,S SAN FRANCISCO,CA 94080
来源
:
CHEMISTRY & BIOLOGY
|
1995年
/ 2卷
/ 12期
关键词
:
D O I
:
10.1016/1074-5521(95)90083-7
中图分类号
:
Q5 [生物化学];
Q7 [分子生物学];
学科分类号
:
071010 ;
081704 ;
摘要
:
引用
收藏
页码:787 / 791
页数:5
相关论文
共 26 条
[1]
CAAX GERANYLGERANYL TRANSFERASE TRANSFERS FARNESYL AS EFFICIENTLY AS GERANYLGERANYL TO RHOB
ARMSTRONG, SA
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
ARMSTRONG, SA
HANNAH, VC
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
HANNAH, VC
GOLDSTEIN, JL
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
GOLDSTEIN, JL
BROWN, MS
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
BROWN, MS
[J].
JOURNAL OF BIOLOGICAL CHEMISTRY,
1995,
270
(14)
: 7864
-
7868
[2]
RAS GENES
BARBACID, M
论文数:
0
引用数:
0
h-index:
0
BARBACID, M
[J].
ANNUAL REVIEW OF BIOCHEMISTRY,
1987,
56
: 779
-
827
[3]
Novel tricyclic inhibitors of farnesyl protein transferase - Biochemical characterization and inhibition of Ras modification in transfected Cos cells
Bishop, WR
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Bishop, WR
Bond, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Bond, R
Petrin, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Petrin, J
Wang, L
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Wang, L
Patton, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Patton, R
Doll, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Doll, R
Njoroge, G
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Njoroge, G
Catino, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Catino, J
Schwartz, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Schwartz, J
Windsor, W
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Windsor, W
Syto, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Syto, R
Schwartz, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Schwartz, J
Carr, D
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Carr, D
James, L
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
James, L
Kirschmeier, P
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Kirschmeier, P
[J].
JOURNAL OF BIOLOGICAL CHEMISTRY,
1995,
270
(51)
: 30611
-
30618
[4]
CARBONI JM, 1995, ONCOGENE, V10, P1905
[5]
FARNESOL IS UTILIZED FOR PROTEIN ISOPRENYLATION AND THE BIOSYNTHESIS OF CHOLESTEROL IN MAMMALIAN-CELLS
CRICK, DC
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
CRICK, DC
ANDRES, DA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
ANDRES, DA
WAECHTER, CJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
WAECHTER, CJ
[J].
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1995,
211
(02)
: 590
-
599
[6]
DALTON MB, 1995, CANCER RES, V55, P3295
[7]
GARCIA AM, 1993, J BIOL CHEM, V268, P18415
[8]
RAS C-TERMINAL PROCESSING ENZYMES - MINIREVIEW NEW DRUG TARGETS
GIBBS, JB
论文数:
0
引用数:
0
h-index:
0
GIBBS, JB
[J].
CELL,
1991,
65
(01)
: 1
-
4
[9]
GIBBS JB, 1993, J BIOL CHEM, V268, P7617
[10]
BENZODIAZEPINE PEPTIDOMIMETICS - POTENT INHIBITORS OF RAS FARNESYLATION IN ANIMAL-CELLS
JAMES, GL
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
JAMES, GL
GOLDSTEIN, JL
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
GOLDSTEIN, JL
BROWN, MS
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
BROWN, MS
RAWSON, TE
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
RAWSON, TE
SOMERS, TC
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
SOMERS, TC
MCDOWELL, RS
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
MCDOWELL, RS
CROWLEY, CW
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
CROWLEY, CW
LUCAS, BK
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
LUCAS, BK
LEVINSON, AD
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
LEVINSON, AD
MARSTERS, JC
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
MARSTERS, JC
[J].
SCIENCE,
1993,
260
(5116)
: 1937
-
1942
←
1
2
3
→
共 26 条
[1]
CAAX GERANYLGERANYL TRANSFERASE TRANSFERS FARNESYL AS EFFICIENTLY AS GERANYLGERANYL TO RHOB
ARMSTRONG, SA
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
ARMSTRONG, SA
HANNAH, VC
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
HANNAH, VC
GOLDSTEIN, JL
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
GOLDSTEIN, JL
BROWN, MS
论文数:
0
引用数:
0
h-index:
0
机构:
Department of Molecular Genetics, Texas University SW Medical Center, Dallas
BROWN, MS
[J].
JOURNAL OF BIOLOGICAL CHEMISTRY,
1995,
270
(14)
: 7864
-
7868
[2]
RAS GENES
BARBACID, M
论文数:
0
引用数:
0
h-index:
0
BARBACID, M
[J].
ANNUAL REVIEW OF BIOCHEMISTRY,
1987,
56
: 779
-
827
[3]
Novel tricyclic inhibitors of farnesyl protein transferase - Biochemical characterization and inhibition of Ras modification in transfected Cos cells
Bishop, WR
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Bishop, WR
Bond, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Bond, R
Petrin, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Petrin, J
Wang, L
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Wang, L
Patton, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Patton, R
Doll, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Doll, R
Njoroge, G
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Njoroge, G
Catino, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Catino, J
Schwartz, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Schwartz, J
Windsor, W
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Windsor, W
Syto, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Syto, R
Schwartz, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Schwartz, J
Carr, D
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Carr, D
James, L
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
James, L
Kirschmeier, P
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Kirschmeier, P
[J].
JOURNAL OF BIOLOGICAL CHEMISTRY,
1995,
270
(51)
: 30611
-
30618
[4]
CARBONI JM, 1995, ONCOGENE, V10, P1905
[5]
FARNESOL IS UTILIZED FOR PROTEIN ISOPRENYLATION AND THE BIOSYNTHESIS OF CHOLESTEROL IN MAMMALIAN-CELLS
CRICK, DC
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
CRICK, DC
ANDRES, DA
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
ANDRES, DA
WAECHTER, CJ
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
UNIV KENTUCKY,COLL MED,MED CTR,DEPT BIOCHEM,LEXINGTON,KY 40536
WAECHTER, CJ
[J].
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS,
1995,
211
(02)
: 590
-
599
[6]
DALTON MB, 1995, CANCER RES, V55, P3295
[7]
GARCIA AM, 1993, J BIOL CHEM, V268, P18415
[8]
RAS C-TERMINAL PROCESSING ENZYMES - MINIREVIEW NEW DRUG TARGETS
GIBBS, JB
论文数:
0
引用数:
0
h-index:
0
GIBBS, JB
[J].
CELL,
1991,
65
(01)
: 1
-
4
[9]
GIBBS JB, 1993, J BIOL CHEM, V268, P7617
[10]
BENZODIAZEPINE PEPTIDOMIMETICS - POTENT INHIBITORS OF RAS FARNESYLATION IN ANIMAL-CELLS
JAMES, GL
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
JAMES, GL
GOLDSTEIN, JL
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
GOLDSTEIN, JL
BROWN, MS
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
BROWN, MS
RAWSON, TE
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
RAWSON, TE
SOMERS, TC
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
SOMERS, TC
MCDOWELL, RS
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
MCDOWELL, RS
CROWLEY, CW
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
CROWLEY, CW
LUCAS, BK
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
LUCAS, BK
LEVINSON, AD
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
LEVINSON, AD
MARSTERS, JC
论文数:
0
引用数:
0
h-index:
0
机构:
GENENTECH INC, DEPT BIOORGAN CHEM, S SAN FRANCISCO, CA 94080 USA
MARSTERS, JC
[J].
SCIENCE,
1993,
260
(5116)
: 1937
-
1942
←
1
2
3
→