REVERSIBLE INHIBITION OF NEURONAL UPTAKE BY BENEXTRAMINE, AN IRREVERSIBLE PRESYNAPTIC ALPHA-ADRENOCEPTOR ANTAGONIST

被引:16
作者
LEW, MJ [1 ]
ANGUS, JA [1 ]
机构
[1] BAKER MED RES INST,COMMERCIAL RD,PRAHRAN,VIC 3181,AUSTRALIA
关键词
D O I
10.1016/0014-2999(84)90105-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:27 / 34
页数:8
相关论文
共 16 条
  • [1] ANGUS JA, 1981, J PHARM METH, V6, P59
  • [2] INHIBITION BY THE TETRAMINE DISULFIDE, BENEXTRAMINE, OF CARDIAC CHRONOTROPIC HISTAMINE H2-RECEPTOR-MEDIATED EFFECTS
    BELLEAU, B
    BENFEY, BG
    BENFEY, TJ
    MELCHIORRE, C
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1982, 75 (04) : 573 - 578
  • [3] PRE-SYNAPTIC EFFECT OF CLONIDINE ANTAGONIZED BY THE TETRAMINE DISULFIDE, BENEXTRAMINE
    BELLEAU, B
    BENFEY, BG
    MELCHIORRE, C
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1982, 75 (04) : 617 - 621
  • [4] IRREVERSIBLE ALPHA-ADRENOCEPTOR BLOCKING EFFECTS AND REVERSIBLE MUSCARINIC BLOCKING AND NICOTINIC BLOCKING EFFECTS OF TETRAMINE DISULFIDES ON THE HEART
    BENFEY, BG
    BELLEAU, B
    BRASILI, L
    GIANNELLA, M
    MELCHIORRE, C
    [J]. CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1980, 58 (12) : 1477 - 1483
  • [5] POTENTIATION AND INHIBITION OF NICOTINIC EFFECTS ON STRIATED-MUSCLE BY THE TETRAMINE DISULFIDE BENEXTRAMINE
    BENFEY, BG
    BRASILI, L
    MELCHIORRE, C
    BELLEAU, B
    [J]. CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1980, 58 (08) : 984 - 988
  • [6] CARDIAC MUSCARINIC BLOCKING AND ATROPINIC BLOCKING EFFECTS OF A TETRAMINE DISULFIDE WITH ALPHA-ADRENOCEPTOR BLOCKING ACTIVITY
    BENFEY, BG
    YONG, MS
    BELLEAU, B
    MELCHIORRE, C
    [J]. CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY, 1979, 57 (01) : 41 - 47
  • [7] BRAZENOR RM, 1981, J PHARMACOL EXP THER, V218, P530
  • [8] FURCHGOTT RF, 1980, VASCULAR NEUROEFFECT
  • [9] DISADVANTAGES OF COCAINE AS A NEURONAL UPTAKE BLOCKING-AGENT - COMPARISON WITH DESIPRAMINE IN GUINEA-PIG RIGHT ATRIUM
    LEW, MJ
    ANGUS, JA
    [J]. JOURNAL OF AUTONOMIC PHARMACOLOGY, 1983, 3 (02): : 61 - 71
  • [10] MOLECULAR-PROPERTIES OF ADRENERGIC ALPHA-RECEPTOR .2. OPTIMUM COVALENT INHIBITION BY 2 DIFFERENT PROTOTYPES OF POLYAMINE DISULFIDES
    MELCHIORRE, C
    YONG, MS
    BENFEY, BG
    BELLEAU, B
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1978, 21 (11) : 1126 - 1132