BINDING OF I-125-LABELED CYANOPINDOLOL TO BETA-1-ADRENOCEPTORS IN A HIGH AND LOW AFFINITY STATE

被引:8
作者
HOYER, D
ENGEL, G
机构
来源
JOURNAL OF RECEPTOR RESEARCH | 1983年 / 3卷 / 1-2期
关键词
D O I
10.3109/10799898309041922
中图分类号
Q2 [细胞生物学];
学科分类号
071009 ; 090102 ;
摘要
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页码:45 / 59
页数:15
相关论文
共 15 条
[1]   BETA-ADRENERGIC-RECEPTOR - STEREOSPECIFIC INTERACTION OF IODINATED BETA-BLOCKING AGENT WITH HIGH AFFINITY SITE [J].
AURBACH, GD ;
FEDAK, SA ;
WOODARD, CJ ;
PALMER, JS .
SCIENCE, 1974, 186 (4170) :1223-1224
[2]  
BEARER CF, 1980, MOL PHARMACOL, V17, P328
[3]  
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[4]  
BURGISSER E, 1981, MOL PHARMACOL, V19, P205
[5]  
DICKINSON KEJ, 1981, BRIT J PHARMACOL, V72, pP165
[6]   (+/)(IODO-125)CYANOPINDOLOL, A NEW LIGAND FOR BETA-ADRENOCEPTORS - IDENTIFICATION AND QUANTITATION OF SUBCLASSES OF BETA-ADRENOCEPTORS IN GUINEA-PIG [J].
ENGEL, G ;
HOYER, D ;
BERTHOLD, R ;
WAGNER, H .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1981, 317 (04) :277-285
[7]   BINDING CHARACTERISTICS OF (+)-, (+/-) AND (-)-[125IODO] CYANOPINDOLOL TO GUINEA-PIG LEFT-VENTRICLE MEMBRANES [J].
HOYER, D ;
ENGEL, G ;
BERTHOLD, R .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 318 (04) :319-329
[8]   BETA-ADRENOCEPTOR BLOCKING-AGENTS AS PARTIAL AGONISTS IN ISOLATED HEART-MUSCLE - DISSOCIATION OF STIMULATION AND BLOCKADE [J].
KAUMANN, AJ ;
BLINKS, JR .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1980, 311 (03) :237-248
[9]  
MAELICKE A, 1977, J BIOL CHEM, V252, P4811
[10]  
POCHET R, 1978, HORMONES CELL REGUL, V2, P133