THE STEREOCONTROLLED SYNTHESIS OF 1,2-CIS FURANOSYL NUCLEOSIDES VIA A NOVEL ANOMERIC ACTIVATION

被引：12

作者：

HANESSIAN, S

CONDE, JJ

LOU, BL

机构：

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 33期

关键词：

D O I：

10.1016/0040-4039(95)01179-L

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The coupling of 2-(2',3',5'-tri-O-benzyl-D-ribofuranosyloxy)-3-methoxypyridine as well as 2-(2',3',5'-tri-O-benzyl-D-ribofuranosyl with silylated pyrimidine bases by activation with trimethylsilyl trifluoromethanesulfonate and silver triflate respectively affords the corresponding 1,2-cis nucleosides with high selectivity.

引用

页码：5865 / 5868

页数：4

共 22 条

[1] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 5-FLUORO-4'-THIOURIDINE AND SOME RELATED NUCLEOSIDES [J].