ALPHA-1-ADRENOCEPTORS - THE ABILITY OF VARIOUS AGONISTS AND ANTAGONISTS TO DISCRIMINATE BETWEEN 2 DISTINCT [H-3]PRAZOSIN BINDING-SITES

被引:49
作者
HANFT, G
GROSS, G
BECKERINGH, JJ
KORSTANJE, C
机构
[1] UNIV ESSEN GESAMTHSCH KLINIKUM,INST PHARMAKOL,HUFELANDSTR 55,D-4300 ESSEN 1,FED REP GER
[2] GIST BROCADES NV RES & DEV,DEPT PHARMACOL,DELFT,NETHERLANDS
关键词
D O I
10.1111/j.2042-7158.1989.tb06348.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:714 / 716
页数:3
相关论文
共 14 条
[1]  
BARLOW RB, 1983, BIODATA HANDLING MIC
[2]   BLOCKADE BY WB 4101 OF ALPHA-ADRENOCEPTORS IN RAT VAS-DEFERENS AND GUINEA-PIG TAENIA CECI [J].
BUTLER, M ;
JENKINSON, DH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 52 (3-4) :303-311
[3]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[4]  
GROSS G, 1988, N-S ARCH PHARMACOL, V338, P582
[5]   5-METHYL-URAPIDIL DISCRIMINATES BETWEEN SUBTYPES OF THE ALPHA-1-ADRENOCEPTOR [J].
GROSS, G ;
HANFT, G ;
RUGEVICS, C .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1988, 151 (02) :333-335
[6]  
HAN C, 1987, MOL PHARMACOL, V32, P505
[7]   ALPHA-1-ADRENOCEPTOR SUBTYPES LINKED TO DIFFERENT MECHANISMS FOR INCREASING INTRACELLULAR CA-2+ IN SMOOTH-MUSCLE [J].
HAN, C ;
ABEL, PW ;
MINNEMAN, KP .
NATURE, 1987, 329 (6137) :333-335
[8]   SUBCLASSIFICATION OF ALPHA-1-ADRENOCEPTOR RECOGNITION SITES BY URAPIDIL DERIVATIVES AND OTHER SELECTIVE ANTAGONISTS [J].
HANFT, G ;
GROSS, G .
BRITISH JOURNAL OF PHARMACOLOGY, 1989, 97 (03) :691-700
[9]  
HIEBLE JP, 1987, ALPHA 1 ADRENERGIC R, P325
[10]  
HONDA K, 1987, N-S ARCH PHARMACOL, V336, P295