CHRONIC ADMINISTRATION OF THE GABA-TRANSAMINASE INHIBITOR ETHANOLAMINE O-SULFATE LEADS TO UP-REGULATION OF GABA BINDING-SITES

被引:29
作者
SYKES, C [1 ]
PRESTWICH, S [1 ]
HORTON, R [1 ]
机构
[1] ST GEORGES HOSP,SCH MED,DEPT PHARMACOL,LONDON SW17 0RE,ENGLAND
关键词
D O I
10.1016/0006-2952(84)90230-2
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:387 / 393
页数:7
相关论文
共 41 条
[1]  
ANLEZARK GM, 1976, BRIT J PHARMACOL, V56, P383
[2]  
BAXTER MG, 1973, BRIT J PHARMACOL, V47, pP681
[3]   HUNTINGTONS-CHOREA - POSTMORTEM MEASUREMENT OF GLUTAMIC-ACID DECARBOXYLASE, CHOLINE-ACETYLTRANSFERASE AND DOPAMINE IN BASAL GANGLIA [J].
BIRD, ED ;
IVERSEN, LL .
BRAIN, 1974, 97 (SEP) :457-472
[4]   CHARACTERISTICS OF GABAB RECEPTOR-BINDING SITES ON RAT WHOLE BRAIN SYNAPTIC-MEMBRANES [J].
BOWERY, NG ;
HILL, DR ;
HUDSON, AL .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 78 (01) :191-206
[5]  
BRENNAN MJW, 1981, MOL PHARMACOL, V19, P27
[6]  
BURCH TP, 1983, MOL PHARMACOL, V23, P52
[7]   ANOREXIC EFFECTS OF ETHANOLAMINE-O-SULFATE AND MUSCIMOL IN THE RAT - EVIDENCE THAT GABA INHIBITS INGESTIVE BEHAVIOR [J].
COOPER, BR ;
HOWARD, JL ;
WHITE, HL ;
SOROKO, F ;
INGOLD, K ;
MAXWELL, RA .
LIFE SCIENCES, 1980, 26 (23) :1997-2002
[8]   MOLECULAR MECHANISMS MEDIATING ACTION OF DIAZEPAM ON GABA RECEPTORS [J].
COSTA, E ;
GUIDOTTI, A ;
TOFFANO, G .
BRITISH JOURNAL OF PSYCHIATRY, 1978, 133 (SEP) :239-248
[9]   RECEPTOR ADAPTATIONS TO CENTRALLY ACTING DRUGS [J].
CREESE, I ;
SIBLEY, DR .
ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1981, 21 :357-391
[10]  
ENNA SJ, 1981, GABA BENZODIAZEPINE, P181