BEHAVIOR OF REACTION MIXTURES UNDER MICROWAVE CONDITIONS - USE OF SODIUM-SALTS IN MICROWAVE-INDUCED N-[F-18]FLUOROALKYLATIONS OF APORPHINE AND TETRALIN DERIVATIVES

被引：34

作者：

ZIJLSTRA, S ^{[1
]}

DEGROOT, TJ ^{[1
]}

KOK, LP ^{[1
]}

VISSER, GM ^{[1
]}

VAALBURG, W ^{[1
]}

机构：

[1] UNIV GRONINGEN,INST THEORET PHYS,9700 AB GRONINGEN,NETHERLANDS

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1993年 / 58卷 / 07期

关键词：

D O I：

10.1021/jo00059a002

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Microwave treatment combined with manipulation of the ionic strength of the reaction mixture increases the radiochemical yield dramatically of N-[F-18]fluoroalkylations of secondary amines as compared to thermal heating.

引用

页码：1643 / 1645

页数：3

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