THE BINDING OF [H-3] LEUKOTRIENE C-4 TO GUINEA-PIG LUNG MEMBRANES - THE LACK OF CORRELATION OF LTC4 FUNCTIONAL-ACTIVITY WITH BINDING-AFFINITY

被引:36
作者
NORMAN, P [1 ]
ABRAM, TS [1 ]
KLUENDER, HC [1 ]
GARDINER, PJ [1 ]
CUTHBERT, NJ [1 ]
机构
[1] MILES LABS INC, ELKHART, IN 46515 USA
关键词
D O I
10.1016/0014-2999(87)90456-0
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:323 / 334
页数:12
相关论文
共 38 条
[1]   INVITRO METABOLISM OF [H-3] PEPTIDE LEUKOTRIENES IN HUMAN AND FERRET LUNG - A COMPARISON WITH THE GUINEA-PIG [J].
AHARONY, D ;
DOBSON, PT ;
KRELL, RD .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1985, 131 (02) :892-898
[2]  
BERENGUER MJ, 1971, TETRAHEDRON LETT, P495
[3]  
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[4]   THE RELEASE OF HISTAMINE AND FORMATION OF A SLOW-REACTING SUBSTANCE (SRS-A) DURING ANAPHYLACTIC SHOCK [J].
BROCKLEHURST, WE .
JOURNAL OF PHYSIOLOGY-LONDON, 1960, 151 (03) :416-435
[5]   ANTIGEN-INDUCED LEUKOTRIENE RELEASE FROM RAT LUNG INVITRO [J].
BRUNET, G ;
CHARLESON, S ;
FORDHUTCHINSON, AW .
PROSTAGLANDINS, 1985, 29 (06) :921-932
[6]   EVIDENCE FOR A SIMILAR RECEPTOR-SITE FOR BINDING OF [H-3] LEUKOTRIENE-E4 AND [H-3] LEUKOTRIENE-D4 TO THE GUINEA-PIG CRUDE LUNG MEMBRANE [J].
CHENG, JB ;
TOWNLEY, RG .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 122 (03) :949-954
[7]   EFFECT OF THE SERINE-BORATE COMPLEX ON THE RELATIVE ABILITY OF LEUKOTRIENE C-4, D4 AND E4 TO INHIBIT LUNG AND BRAIN [H-3] LEUKOTRIENE-D4 AND [H-3] LEUKOTRIENE-C4 BINDING - DEMONSTRATION OF THE AGONISTS POTENCY ORDER FOR LEUKOTRIENE-D4 AND LEUKOTRIENE-C4 RECEPTORS [J].
CHENG, JB ;
TOWNLEY, RG .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 119 (02) :612-617
[8]  
CHENG Y, 1973, BIOCHEM PHARMACOL, V22, P3099
[9]  
COOPER DMF, 1983, CURR TOP MEMBR TRANS, V18, P67
[10]  
CUTHBERT NJ, 1987, BRIT J PHARMACOL, pP408