A MINOR MODIFICATION OF RESIDUE 1 IN POTENT VASOPRESSIN ANTAGONISTS DRAMATICALLY REDUCES AGONIST ACTIVITY

[1] ALBRIGHTSON C, 1987, FED PROC, V46, P1284

[2] POTENT VASOPRESSIN ANTAGONISTS MODIFIED AT THE CARBOXY-TERMINAL TRIPEPTIDE TAIL [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (12) : 2291 - 2294

[3] POTENT VASOPRESSIN ANTAGONISTS LACKING THE PROLINE RESIDUE AT POSITION-7 [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (06) : 984 - 988

[4] ARIENS EJ, 1979, RECEPTORS, V1, pCH2

[5] MOLECULAR THEORY OF DRUG ACTION BASED ON INDUCED CONFORMATIONAL PERTURBATIONS OF RECEPTORS [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1964, 7 (06) : 776 - &

[6] AN IMPROVED PREPARATION OF BENZHYDRYLAMINE RESIN [J]. JOURNAL OF ORGANIC CHEMISTRY, 1986, 51 (17) : 3371 - 3372

[7] Carman-Krzan M, 1986, Prog Med Chem, V23, P41, DOI 10.1016/S0079-6468(08)70340-0

[8] DEBROSSE CW, 1988, PEPTIDES CHEM BIOL, P68

[9] DUBB J, 1987, KIDNEY INT, V31, P267

[10] EGGLESTON DS, IN PRESS ACTA CRYSTA

[1] ALBRIGHTSON C, 1987, FED PROC, V46, P1284

[2] POTENT VASOPRESSIN ANTAGONISTS MODIFIED AT THE CARBOXY-TERMINAL TRIPEPTIDE TAIL [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (12) : 2291 - 2294

[3] POTENT VASOPRESSIN ANTAGONISTS LACKING THE PROLINE RESIDUE AT POSITION-7 [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1986, 29 (06) : 984 - 988

[4] ARIENS EJ, 1979, RECEPTORS, V1, pCH2

[5] MOLECULAR THEORY OF DRUG ACTION BASED ON INDUCED CONFORMATIONAL PERTURBATIONS OF RECEPTORS [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1964, 7 (06) : 776 - &

[6] AN IMPROVED PREPARATION OF BENZHYDRYLAMINE RESIN [J]. JOURNAL OF ORGANIC CHEMISTRY, 1986, 51 (17) : 3371 - 3372

[7] Carman-Krzan M, 1986, Prog Med Chem, V23, P41, DOI 10.1016/S0079-6468(08)70340-0

[8] DEBROSSE CW, 1988, PEPTIDES CHEM BIOL, P68

[9] DUBB J, 1987, KIDNEY INT, V31, P267

[10] EGGLESTON DS, IN PRESS ACTA CRYSTA