SYNTHESIS OF A NEW TETRACYCLIC SYSTEM RELATED TO APTAZAPINE (CGS-7525A) BY ONE-POT DOUBLE ANNELATION

被引：14

作者：

MASSA, S ^{[1
]}

MAI, A ^{[1
]}

CORELLI, F ^{[1
]}

机构：

[1] DIPARTIMENTO FARM CHIM TECHNOL, I-53100 SIENA, ITALY

来源：

TETRAHEDRON LETTERS | 1988年 / 29卷 / 49期

关键词：

D O I：

10.1016/S0040-4039(00)82376-X

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：6471 / 6474

页数：4

共 10 条

[1]

Ankier S I, 1986, Prog Med Chem, V23, P121, DOI 10.1016/S0079-6468(08)70342-4

[2] INHIBITION OF COPPER-DEPENDENT AMINE OXIDASES BY SOME HYDRAZIDES OF PYRROL-1-YLBENZOIC AND PYRROL-1-YLPHENYLACETIC ACIDS [J].

ARTICO, M ;

CORELLI, F ;

MASSA, S ;

STEFANCICH, G ;

AVIGLIANO, L ;

BEFANI, O ;

MARCOZZI, G ;

SABATINI, S ;

MONDOVI, B .

JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (04) :802-806

[3] A PRACTICAL SYNTHESIS OF 1,3,4,14B-TETRAHYDRO-2-METHYL-10H-PYRAZINO[1,2-A]PYRROLO[2,1-C][1,4]BENZODIAZEPINE (1-1) MALEATE [J].

BOYER, SK ;

FITCHETT, G ;

WASLEY, JWF ;

ZAUNIUS, G .

JOURNAL OF HETEROCYCLIC CHEMISTRY, 1984, 21 (03) :833-835

[4] FURTHER CYCLISATION REACTIONS OF 1-ARYLPYRROLES [J].

CHEESEMAN, GW ;

RAFIQ, M .

JOURNAL OF THE CHEMICAL SOCIETY C-ORGANIC, 1971, (15) :2732-+

[5]

CORELLI F, 1986, EUR J MED CHEM, V21, P445

[6]

KANO S, 1984, SYNTHESIS-STUTTGART, P1071

[7] PYRROLOISOQUINOLINE ANTIDEPRESSANTS .2. IN-DEPTH EXPLORATION OF STRUCTURE-ACTIVITY-RELATIONSHIPS [J].

MARYANOFF, BE ;

MCCOMSEY, DF ;

GARDOCKI, JF ;

SHANK, RP ;

COSTANZO, MJ ;

NORTEY, SO ;

SCHNEIDER, CR ;

SETLER, PE .

JOURNAL OF MEDICINAL CHEMISTRY, 1987, 30 (08) :1433-1454

[8]

MASSA S, 1985, HETEROCYCLES, V23, P1417

[9] ATYPICAL ANTIPSYCHOTIC AGENTS - PATTERNS OF ACTIVITY IN A SERIES OF 3-SUBSTITUTED 2-PYRIDINYL-1-PIPERAZINE DERIVATIVES [J].

NEW, JS ;

YEVICH, JP ;

TEMPLE, DL ;

NEW, KB ;

GROSS, SM ;

SCHLEMMER, RF ;

EISON, MS ;

TAYLOR, DP ;

RIBLET, LA .

JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (03) :618-624

[10] SYNTHESIS AND BIOLOGICAL PROPERTIES OF THIOPHENE RING ANALOGS OF MIANSERIN [J].

WATTHEY, JWH ;

GAVIN, T ;

DESAI, M ;

FINN, BM ;

RODEBAUGH, RK ;

PATT, SL .

JOURNAL OF MEDICINAL CHEMISTRY, 1983, 26 (08) :1116-1122

← 1 →