QUATERNARY DERIVATIVES OF NARCOTIC-ANTAGONISTS - STEREOCHEMICAL REQUIREMENTS AT THE CHIRAL NITROGEN FOR INVITRO AND INVIVO ACTIVITY

被引：19

作者：

BIANCHETTI, A ^{[1
]}

NISATO, D ^{[1
]}

SACILOTTO, R ^{[1
]}

DRAGONETTI, M ^{[1
]}

PICERNO, N ^{[1
]}

TARANTINO, A ^{[1
]}

MANARA, L ^{[1
]}

ANGEL, LM ^{[1
]}

SIMON, EJ ^{[1
]}

机构：

[1] NYU,SCH MED,DEPT PSYCHIAT & PHARMACOL,NEW YORK,NY 10016

来源：

LIFE SCIENCES | 1983年 / 33卷

关键词：

D O I：

10.1016/0024-3205(83)90530-1

中图分类号：

R-3 [医学研究方法]; R3 [基础医学];

学科分类号：

1001 ;

摘要：

引用

页码：415 / 418

页数：4

共 10 条

[1] PHARMACOLOGICAL ACTIONS OF LEVALLORPHAN ALLYL BROMIDE (CM-32191), A NEW PERIPHERAL NARCOTIC-ANTAGONIST
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[J]. LIFE SCIENCES, 1982, 31 (20-2) : 2261 - 2264
[2] QUATERNARY NARCOTIC-ANTAGONISTS RELATIVE ABILITY TO PREVENT ANTINOCICEPTION AND GASTROINTESTINAL TRANSIT INHIBITION IN MORPHINE-TREATED RATS AS AN INDEX OF PERIPHERAL SELECTIVITY
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[J]. LIFE SCIENCES, 1982, 30 (22) : 1875 - 1883
[3] EFFECTS OF NALOXONE AND ITS QUATERNARY ANALOG ON STIMULATION-INDUCED FEEDING
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[J]. NEUROPHARMACOLOGY, 1983, 22 (01) : 127 - 130
[4] DRAGONETTI M, 1983, LIFE SCI S1, V33
[5] OPIATE RECEPTOR - MODEL EXPLAINING STRUCTURE-ACTIVITY-RELATIONSHIPS OF OPIATE AGONISTS AND ANTAGONISTS
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[6] N-METHYLNALORPHINE - DEFINITION OF N-ALLYL CONFORMATION FOR ANTAGONISM AT THE OPIATE RECEPTOR
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[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1982, 25 (11) : 1278 - 1280
[7] KOCZKA K, 1967, ACTA CHIM HUNG, V51, P393
[8] KINETIC PARAMETERS OF NARCOTIC AGONISTS AND ANTAGONISTS WITH PARTICULAR REFERENCE TO N-ALLYLNOROXYMORPHONE (NALOXONE)
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WATT, AJ
[J]. BRITISH JOURNAL OF PHARMACOLOGY, 1968, 33 (02) : 266 - +
[9] INVITRO MODELS IN STUDY OF STRUCTURE-ACTIVITY-RELATIONSHIPS OF NARCOTIC ANALGESICS
KOSTERLITZ, HW
WATERFIELD, AA
[J]. ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY, 1975, 15 : 29 - 47
[10] SIMON EJ, 1975, J PHARMACOL EXP THER, V192, P531

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