THE INFLUENCE OF SELECTIVE THROMBOXANE SYNTHETASE INHIBITION WITH A NOVEL IMIDAZOLE DERIVATIVE, UK-38,485, ON PROSTANOID FORMATION IN MAN

被引:93
作者
FISCHER, S
STRUPPLER, M
BOHLIG, B
BERNUTZ, C
WOBER, W
WEBER, PC
机构
[1] UNIV MUNICH, MED KLIN INNENSTADT, D-8000 MUNICH 2, FED REP GER
[2] PFIZER CLIN RES, MUNCHEN, FED REP GER
关键词
D O I
10.1161/01.CIR.68.4.821
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页码:821 / 826
页数:6
相关论文
共 25 条
[1]  
AIKEN JW, 1981, J PHARMACOL EXP THER, V219, P299
[2]   A THROMBOXANE SYNTHETASE INHIBITOR RE-ORIENTS ENDOPEROXIDE METABOLISM IN WHOLE-BLOOD TOWARDS PROSTACYCLIN AND PROSTAGLANDIN-E2 [J].
DEFREYN, G ;
DECKMYN, H ;
VERMYLEN, J .
THROMBOSIS RESEARCH, 1982, 26 (06) :389-400
[3]   QUANTITATIVE ANALYSIS OF TWO DINOR URINARY METABOLITES OF PROSTAGLANDIN I2 [J].
FALARDEAU, P ;
OATES, JA ;
BRASH, AR .
ANALYTICAL BIOCHEMISTRY, 1981, 115 (02) :359-367
[4]   PROSTACYCLIN METABOLISM IN ADULTS AND NEONATES - URINARY PROFILES OF 6-KETOPROSTAGLANDIN-F1-ALPHA AND 2,3-DINOR-6-KETOPROSTAGLANDIN-F1-ALPHA STUDIED BY GAS CHROMATOGRAPHY-MASS SPECTROMETRY [J].
FISCHER, S ;
SCHERER, B ;
WEBER, PC .
BIOCHIMICA ET BIOPHYSICA ACTA, 1983, 750 (01) :127-133
[5]  
FOEGH ML, 1981, LANCET, V2, P431
[6]  
Harris D N, 1980, Adv Prostaglandin Thromboxane Res, V6, P437
[7]   CONTRIBUTION OF THROMBOXANE TO RENAL RESISTANCE CHANGES IN THE ISOLATED PERFUSED HYDRONEPHROTIC RABBIT KIDNEY [J].
KAWASAKI, A ;
NEEDLEMAN, P .
CIRCULATION RESEARCH, 1982, 50 (04) :486-490
[8]  
LEWY R I, 1979, Clinical Cardiology, V2, P404
[9]  
McGuire J C, 1980, Adv Prostaglandin Thromboxane Res, V8, P1665
[10]   UNSTABLE METABOLITES OF ARACHIDONIC-ACID AND THEIR ROLE IN HEMOSTASIS AND THROMBOSIS [J].
MONCADA, S ;
VANE, JR .
BRITISH MEDICAL BULLETIN, 1978, 34 (02) :129-135