SYNTHESIS OF PYRROLO[1,2-C]QUINAZOLINE DERIVATIVES

被引：11

作者：

BECCALLI, EM

MARCHESINI, A

PILATI, T

机构：

[1] UNIV MILAN,DIPARTIMENTO CHIM ORGAN & IND,VIA GOLGI 19,I-20133 MILAN,ITALY

[2] CNR,CTR STUDIO RELAZIONI STRUTTURA & REATTIVITA CHIM,I-20133 MILAN,ITALY

来源：

TETRAHEDRON | 1992年 / 48卷 / 25期

关键词：

2H-INDOL-2-ONES; DELTA-2-PYRROLIN-4-ONES; PYRROLO[1,2-C]QUINAZOLINES;

D O I：

10.1016/S0040-4020(01)89032-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

DELTA-2-Pyrrolin-4-ones 12 and 13, prepared from 1-acyl-3-alkyl-1,3-dihydro-2H-indol-2-ones 1, via the corresponding 3-bromo-, 2 and 6,3-azido, 7 and 8, and 3-iminophosphorane 9 and 10, were cyclized to the corresponding pyrrolo[1,2-c]quinazoline derivatives 14 and 15.

引用

页码：5359 / 5374

页数：16

共 15 条

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[8]

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[9]

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[10]

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