PHARMACOKINETIC PHARMACODYNAMIC ANALYSIS OF UNBOUND DISOPYRAMIDE DIRECTLY MEASURED IN SERIAL PLASMA SAMPLES IN MAN

被引:41
作者
THIBONNIER, M [1 ]
HOLFORD, NHG [1 ]
UPTON, RA [1 ]
BLUME, CD [1 ]
WILLIAMS, RL [1 ]
机构
[1] UNIV CALIF SAN FRANCISCO,SCH PHARM,SAN FRANCISCO,CA 94143
来源
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS | 1984年 / 12卷 / 06期
关键词
D O I
10.1007/BF01059552
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:559 / 573
页数:15
相关论文
共 26 条
[1]  
AITO ML, 1981, BR J CLIN PHARM, V11, P369
[2]  
BRADFORD MM, 1976, ANAL BIOCHEM, V72, P248, DOI 10.1016/0003-2697(76)90527-3
[3]   DISOPYRAMIDE SERUM AND PHARMACOLOGIC EFFECT KINETICS APPLIED TO ASSESSMENT OF BIOAVAILABILITY [J].
BRYSON, SM ;
WHITING, B ;
LAWRENCE, JR .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1978, 6 (05) :409-419
[4]   THE INFLUENCE OF PROTEIN-BINDING ON DISOPYRAMIDE CLEARANCE [J].
BRYSON, SM ;
LAWRENCE, JR ;
STEELE, WH ;
CAMPBELL, BC ;
ELLIOTT, HL ;
SUMNER, DJ .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1982, 23 (05) :453-456
[5]   EFFECTS OF URINE PH AND PLASMA-PROTEIN BINDING ON RENAL CLEARANCE OF DISOPYRAMIDE [J].
CUNNINGHAM, JL ;
SHEN, DD ;
SHUDO, I ;
AZARNOFF, DL .
CLINICAL PHARMACOKINETICS, 1977, 2 (05) :373-383
[6]   PLASMA-BINDING OF DISOPYRAMIDE [J].
DAVID, BM ;
MADSEN, BW ;
ILETT, KF .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1980, 9 (06) :614-618
[7]   THE EFFECT OF SATURABLE BINDING TO PLASMA-PROTEINS ON THE PHARMACOKINETIC PROPERTIES OF DISOPYRAMIDE [J].
GIACOMINI, KM ;
SWEZEY, SE ;
TURNERTAMIYASU, K ;
BLASCHKE, TF .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1982, 10 (01) :1-14
[8]   PROTEIN-BINDING AND ERYTHROCYTE PARTITIONING OF DISOPYRAMIDE AND ITS MONODEALKYLATED METABOLITE [J].
HINDERLING, PH ;
BRES, J ;
GARRETT, ER .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1974, 63 (11) :1684-1690
[9]   PHARMACOKINETICS OF ANTIARRHYTHMIC DISOPYRAMIDE IN HEALTHY HUMANS [J].
HINDERLING, PH ;
GARRETT, ER .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1976, 4 (03) :199-230
[10]  
HOLFORD NHG, 1983, CLIN PHARMACOL THER, V33, P201