A PROTECTION SCHEME FOR THE PREPARATION OF ACID-CHLORIDES OF SERINE AND THREONINE

被引：28

作者：

XI, N ^{[1
]}

CIUFOLINI, MA ^{[1
]}

机构：

[1] RICE UNIV,DEPT CHEM,HOUSTON,TX 77251

来源：

TETRAHEDRON LETTERS | 1995年 / 36卷 / 37期

关键词：

D O I：

10.1016/00404-0399(50)1348-L

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

N-acetyl oxazolone derivatives of serine and threonine are readily converted into reactive acid chlorides that condense efficiently with various C-protected aminoacids, even poorly nucleophilic ones.

引用

页码：6595 / 6598

页数：4

共 17 条

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