STAUROSPORINE, K-252 AND UCN-01 - POTENT BUT NONSPECIFIC INHIBITORS OF PROTEIN-KINASES

被引:974
作者
RUEGG, UT [1 ]
BURGESS, GM [1 ]
机构
[1] UCL, SANDOZ INST MED RES, LONDON WC1E 6BN, ENGLAND
关键词
D O I
10.1016/0165-6147(89)90263-0
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:218 / 220
页数:3
相关论文
共 32 条
[1]  
BURGESS GM, 1988, J PHYSIOL-LONDON, V398, pP17
[2]  
BURGESS GM, IN PRESS J NEUROSCI
[3]  
CHENG HC, 1986, J BIOL CHEM, V261, P989
[4]   BRADYKININ-INDUCED STIMULATION OF AFFERENT-FIBERS IS MEDIATED THROUGH PROTEIN KINASE-C [J].
DRAY, A ;
BETTANEY, J ;
FORSTER, P ;
PERKINS, MN .
NEUROSCIENCE LETTERS, 1988, 91 (03) :301-307
[5]   PROTEIN SERINE THREONINE KINASES [J].
EDELMAN, AM ;
BLUMENTHAL, DK ;
KREBS, EG .
ANNUAL REVIEW OF BIOCHEMISTRY, 1987, 56 :567-613
[6]   PHORBOL ESTER INCREASES THE DIHYDROPYRIDINE-SENSITIVE CALCIUM CONDUCTANCE IN A VASCULAR SMOOTH-MUSCLE CELL-LINE [J].
FISH, RD ;
SPERTI, G ;
COLUCCI, WS ;
CLAPHAM, DE .
CIRCULATION RESEARCH, 1988, 62 (05) :1049-1054
[7]  
GALIZZI JP, 1987, J BIOL CHEM, V262, P6947
[8]   RECEPTOR-MEDIATED CA-2+ ENTRY - DIVERSITY OF FUNCTION AND MECHANISM [J].
HALLAM, TJ ;
RINK, TJ .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1989, 10 (01) :8-10
[9]   THE PROTEIN-KINASE FAMILY - CONSERVED FEATURES AND DEDUCED PHYLOGENY OF THE CATALYTIC DOMAINS [J].
HANKS, SK ;
QUINN, AM ;
HUNTER, T .
SCIENCE, 1988, 241 (4861) :42-52
[10]   ISOQUINOLINESULFONAMIDES, NOVEL AND POTENT INHIBITORS OF CYCLIC-NUCLEOTIDE DEPENDENT PROTEIN-KINASE AND PROTEIN KINASE-C [J].
HIDAKA, H ;
INAGAKI, M ;
KAWAMOTO, S ;
SASAKI, Y .
BIOCHEMISTRY, 1984, 23 (21) :5036-5041