CONFORMATIONALLY CONSTRAINED CYCLIC ENKEPHALIN ANALOGS WITH PRONOUNCED DELTA-OPIOID RECEPTOR AGONIST SELECTIVITY

被引：98

作者：

MOSBERG, HI

HURST, R

HRUBY, VJ

GALLIGAN, JJ

BURKS, TF

GEE, K

YAMAMURA, HI

机构：

[1] UNIV ARIZONA,DEPT BIOCHEM,TUCSON,AZ 85721

[2] UNIV ARIZONA,DEPT PHARMACOL,TUCSON,AZ 85721

来源：

LIFE SCIENCES | 1983年 / 32卷 / 22期

关键词：

D O I：

10.1016/0024-3205(83)90239-4

中图分类号：

R-3 [医学研究方法]; R3 [基础医学];

学科分类号：

1001 ;

摘要：

引用

页码：2565 / 2569

页数：5

共 15 条

[1]

BEDELL C, 1977, P ROY SOC LOND B BIO, V198, P249

[2]

CHANG KJ, 1979, J BIOL CHEM, V254, P2610

[3] MULTIPLE OPIATE RECEPTORS [J].

CHANG, KJ ;

HAZUM, E ;

CUATRECASAS, P .

TRENDS IN NEUROSCIENCES, 1980, 3 (07) :160-162

[4] A CYCLIC ENKEPHALIN ANALOG WITH HIGH INVITRO OPIATE ACTIVITY [J].

DIMAIO, J ;

SCHILLER, PW .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (12) :7162-7166

[5]

FOURNIEZALUSKI MC, 1981, MOL PHARMACOL, V20, P484

[6] CONFORMATIONAL AND DYNAMIC CONSIDERATIONS IN PEPTIDE STRUCTURE-FUNCTION STUDIES [J].

HRUBY, VJ ;

MOSBERG, HI .

PEPTIDES, 1982, 3 (03) :329-336

[7]

HRUBY VJ, 1982, HORMONE ANTAGONISTS, P433

[8] EFFECT OF MORPHINE ON ADRENERGIC TRANSMISSION IN MOUSE VAS-DEFERENS ASSESSMENT OF AGONIST AND ANTAGONIST POTENCIES OF NARCOTIC ANALGESICS [J].

HUGHES, J ;

KOSTERLITZ, HW ;

LESLIE, FM .

BRITISH JOURNAL OF PHARMACOLOGY, 1975, 53 (03) :371-381

[9] EFFECTS OF ADRENALINE, NORADRENALINE AND ISOPRENALINE ON INHIBITORY ALPHA-AND BETA-ADRENOCEPTORS IN LONGITUDINAL MUSCLE OF GUINEA-PIG ILEUM [J].

KOSTERLITZ, HW ;

LYDON, RJ ;

WATT, AJ .

BRITISH JOURNAL OF PHARMACOLOGY, 1970, 39 (02) :398-+

[10] EFFECTS OF CHANGES IN THE STRUCTURE OF ENKEPHALINS AND OF NARCOTIC ANALGESIC DRUGS ON THEIR INTERACTIONS WITH MU-RECEPTOR AND DELTA-RECEPTOR [J].

KOSTERLITZ, HW ;

LORD, JAH ;

PATERSON, SJ ;

WATERFIELD, AA .

BRITISH JOURNAL OF PHARMACOLOGY, 1980, 68 (02) :333-342

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