KINETICS OF CHOLINESTERASE INHIBITION BY EPTASTIGMINE IN MAN

被引:36
作者
UNNI, LK
HUTT, V
IMBIMBO, BP
BECKER, RE
机构
[1] MEDIOLANUM FARMACEUT,DEPT MED,VIA C COLOMBO 49,I-20090 TREZZANO S-N,ITALY
[2] SO ILLINOIS UNIV,SCH MED,DEPT PSYCHIAT,NEUROCHEM LAB,SPRINGFIELD,IL 62708
[3] LAB,DEPT PHASE 1,NEU ULM,GERMANY
关键词
EPTASTIGMINE; CHOLINESTERASE INHIBITOR; ALZHEIMERS DISEASE; PHARMACOKINETICS; ADVERSE EFFECTS;
D O I
10.1007/BF00280116
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:83 / 84
页数:2
相关论文
共 15 条
[1]   MECHANISMS OF CHOLINESTERASE INHIBITION IN SENILE DEMENTIA OF THE ALZHEIMER TYPE - CLINICAL, PHARMACOLOGICAL, AND THERAPEUTIC ASPECTS [J].
BECKER, RE ;
GIACOBINI, E .
DRUG DEVELOPMENT RESEARCH, 1988, 12 (3-4) :163-195
[2]   EFFECTS OF METRIFONATE, A LONG-ACTING CHOLINESTERASE INHIBITOR, IN ALZHEIMER-DISEASE - REPORT OF AN OPEN TRIAL [J].
BECKER, RE ;
COLLIVER, J ;
ELBLE, R ;
FELDMAN, E ;
GIACOBINI, E ;
KUMAR, V ;
MARKWELL, S ;
MORIEARTY, P ;
PARKS, R ;
SHILLCUTT, SD ;
UNNI, L ;
VICARI, S ;
WOMACK, C ;
ZEC, RF .
DRUG DEVELOPMENT RESEARCH, 1990, 19 (04) :425-434
[3]   ANTICHOLINESTERASE ACTIVITY OF A NEW CARBAMATE, HEPTYLPHYSOSTIGMINE, IN VIEW OF ITS USE IN PATIENTS WITH ALZHEIMER-TYPE DEMENTIA [J].
BRUFANI, M ;
MARTA, M ;
POMPONI, M .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1986, 157 (01) :115-120
[4]   A LONG-LASTING CHOLINESTERASE INHIBITOR AFFECTING NEURAL AND BEHAVIORAL PROCESSES [J].
BRUFANI, M ;
CASTELLANO, C ;
MARTA, M ;
OLIVERIO, A ;
PAGELLA, PG ;
PAVONE, F ;
POMPONI, M ;
RUGARLI, PL .
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1987, 26 (03) :625-629
[5]  
DAVIS KL, 1982, AM J PSYCHIAT, V139, P1421
[6]   THE EFFECT OF HEPTYL-PHYSOSTIGMINE, A NEW CHOLINESTERASE INHIBITOR, ON THE CENTRAL CHOLINERGIC SYSTEM OF THE RAT [J].
DESARNO, P ;
POMPONI, M ;
GIACOBINI, E ;
TANG, XC ;
WILLIAMS, E .
NEUROCHEMICAL RESEARCH, 1989, 14 (10) :971-977
[7]   RAPID, SIMPLE RADIOMETRIC ASSAY FOR CHOLINESTERASE, SUITABLE FOR MULTIPLE DETERMINATIONS [J].
JOHNSON, CD ;
RUSSELL, RL .
ANALYTICAL BIOCHEMISTRY, 1975, 64 (01) :229-238
[8]   EXTRACTION OF PHYSOSTIGMINE FROM BIOLOGIC FLUIDS AND ANALYSIS BY LIQUID-CHROMATOGRAPHY WITH ELECTROCHEMICAL DETECTION [J].
LAWRENCE, GD ;
YATIM, N .
JOURNAL OF PHARMACOLOGICAL METHODS, 1990, 24 (02) :137-143
[9]   NEW ANALOGS OF PHYSOSTIGMINE - ALTERNATIVE DRUGS FOR ALZHEIMERS-DISEASE [J].
MARTA, M ;
CASTELLANO, C ;
OLIVERIO, A ;
PAVONE, F ;
PAGELLA, PG ;
BRUFANI, M ;
POMPONI, M .
LIFE SCIENCES, 1988, 43 (23) :1921-1928
[10]  
OLIVERIO A, 1986, MODULATION CENTRAL P, P305