PHARMACOLOGICAL EVIDENCE FOR THE INVOLVEMENT OF ALPHA-2 ADRENOCEPTORS IN THE SEDATIVE EFFECT OF DETOMIDINE, A NOVEL SEDATIVE-ANALGESIC

被引:53
作者
VIRTANEN, R [1 ]
RUSKOAHO, H [1 ]
NYMAN, L [1 ]
机构
[1] UNIV OULU,DEPT PHARMACOL,SF-90100 OULU 10,FINLAND
关键词
D O I
10.1111/j.1365-2885.1985.tb00921.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:30 / 37
页数:8
相关论文
共 17 条
[1]   THE PHYSIOLOGICAL-ROLE OF ALPHA-ADRENOCEPTORS IN THE CNS - NEW CONCEPTS FROM SINGLE-CELL STUDIES [J].
AGHAJANIAN, GK ;
ROGAWSKI, MA .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1983, 4 (07) :315-317
[2]   XYLAZINE - A NEW SEDATIVE FOR HORSES AND CATTLE [J].
CLARKE, KW ;
HALL, LW .
VETERINARY RECORD, 1969, 85 (19) :512-&
[3]   HYPOTENSIVE AND SEDATIVE EFFECTS OF ALPHA-ADRENOCEPTOR AGONISTS - RELATIONSHIP TO ALPHA-1-ADRENOCEPTOR AND ALPHA-2-ADRENOCEPTOR POTENCY [J].
CLOUGH, DP ;
HATTON, R .
BRITISH JOURNAL OF PHARMACOLOGY, 1981, 73 (03) :595-604
[4]   SEDATIVE EFFECTS OF ALPHA-SYMPATHOMIMETIC DRUGS AND THEIR ANTAGONISM BY ADRENERGIC AND CHOLINERGIC BLOCKING DRUGS [J].
DELBARRE, B ;
SCHMITT, H .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1971, 13 (03) :356-&
[5]   DEPRESSION OF EXPLORATORY ACTIVITY BY CLONIDINE IN RATS AS A MODEL FOR THE DETECTION OF RELATIVE PRESYNAPTIC AND POSTSYNAPTIC CENTRAL NORADRENERGIC RECEPTOR SELECTIVITY OF ALPHA-ADRENOLYTIC DRUGS [J].
DELINISTULA, A ;
BAUMANN, P ;
BUCH, O .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1979, 307 (02) :115-122
[6]   STUDIES ON RX781094 - A SELECTIVE, POTENT AND SPECIFIC ANTAGONIST OF ALPHA-2-ADRENOCEPTORS [J].
DOXEY, JC ;
ROACH, AG ;
SMITH, CFC .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 78 (03) :489-505
[7]  
HSU WH, 1981, J PHARMACOL EXP THER, V218, P188
[8]  
KERR DD, 1972, AM J VET RES, V33, P525
[9]   PRESYNAPTIC RECEPTORS AND THEIR ROLE IN REGULATION OF TRANSMITTER RELEASE [J].
LANGER, SZ .
BRITISH JOURNAL OF PHARMACOLOGY, 1977, 60 (04) :481-497
[10]  
LOWRY OH, 1951, J BIOL CHEM, V193, P265