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PHARMACOKINETICS OF MORPHINE AND ITS SURROGATES .6. BIOANALYSIS, SOLVOLYSIS KINETICS, SOLUBILITY, PK'A VALUES, AND PROTEIN-BINDING OF BUPRENORPHINE
被引:36
作者
:
GARRETT, ER
论文数:
0
引用数:
0
h-index:
0
GARRETT, ER
CHANDRAN, VR
论文数:
0
引用数:
0
h-index:
0
CHANDRAN, VR
机构
:
来源
:
JOURNAL OF PHARMACEUTICAL SCIENCES
|
1985年
/ 74卷
/ 05期
关键词
:
D O I
:
10.1002/jps.2600740505
中图分类号
:
R914 [药物化学];
学科分类号
:
100701 ;
摘要
:
引用
收藏
页码:515 / 524
页数:10
相关论文
共 35 条
[1]
THE RADIOIMMUNOASSAY OF BUPRENORPHINE
[J].
BARTLETT, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
BARTLETT, AJ
;
LLOYDJONES, JG
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
LLOYDJONES, JG
;
RANCE, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
RANCE, MJ
;
FLOCKHART, IR
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
FLOCKHART, IR
;
DOCKRAY, GJ
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
DOCKRAY, GJ
;
BENNETT, MRD
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
BENNETT, MRD
;
MOORE, RA
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
MOORE, RA
.
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY,
1980,
18
(04)
:339
-345
[2]
SUB-LINGUAL BUPRENORPHINE USED POSTOPERATIVELY - 10-HOUR PLASMA DRUG CONCENTRATION ANALYSIS
[J].
BULLINGHAM, RES
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
BULLINGHAM, RES
;
MCQUAY, HJ
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
MCQUAY, HJ
;
PORTER, EJB
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
PORTER, EJB
;
ALLEN, MC
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
ALLEN, MC
;
MOORE, RA
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
MOORE, RA
.
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY,
1982,
13
(05)
:665
-673
[3]
AN ORAL BUPRENORPHINE AND PARACETAMOL COMBINATION COMPARED WITH PARACETAMOL ALONE - A SINGLE DOSE DOUBLE-BLIND POSTOPERATIVE STUDY
[J].
BULLINGHAM, RES
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
BULLINGHAM, RES
;
MCQUAY, HJ
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
MCQUAY, HJ
;
MOORE, RA
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
MOORE, RA
;
WEIR, L
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
WEIR, L
.
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY,
1981,
12
(06)
:863
-867
[4]
BUPRENORPHINE KINETICS
[J].
BULLINGHAM, RES
论文数:
0
引用数:
0
h-index:
0
机构:
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
BULLINGHAM, RES
;
MCQUAY, HJ
论文数:
0
引用数:
0
h-index:
0
机构:
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
MCQUAY, HJ
;
MOORE, A
论文数:
0
引用数:
0
h-index:
0
机构:
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
MOORE, A
;
BENNETT, MRD
论文数:
0
引用数:
0
h-index:
0
机构:
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
BENNETT, MRD
.
CLINICAL PHARMACOLOGY & THERAPEUTICS,
1980,
28
(05)
:667
-672
[5]
COMPARISON OF BUPRENORPHINE AND PETHIDINE GIVEN INTRAVENOUSLY ON DEMAND TO RELIEVE POST-OPERATIVE PAIN
[J].
CHAKRAVARTY, K
论文数:
0
引用数:
0
h-index:
0
机构:
Jipmer, Pondicherry
CHAKRAVARTY, K
;
TUCKER, W
论文数:
0
引用数:
0
h-index:
0
机构:
Jipmer, Pondicherry
TUCKER, W
;
ROSEN, M
论文数:
0
引用数:
0
h-index:
0
机构:
Jipmer, Pondicherry
ROSEN, M
;
VICKERS, MD
论文数:
0
引用数:
0
h-index:
0
机构:
Jipmer, Pondicherry
VICKERS, MD
.
BRITISH MEDICAL JOURNAL,
1979,
2
(6195)
:895
-897
[6]
STABILITY OF THE "6,14-ENDO-ETHANOTETRAHYDROORIPAVINE ANALGESICS - ACID-CATALYZED REARRANGEMENT OF BUPRENORPHINE
[J].
CONE, EJ
论文数:
0
引用数:
0
h-index:
0
CONE, EJ
;
GORODETZKY, CW
论文数:
0
引用数:
0
h-index:
0
GORODETZKY, CW
;
DARWIN, WD
论文数:
0
引用数:
0
h-index:
0
DARWIN, WD
;
BUCHWALD, WF
论文数:
0
引用数:
0
h-index:
0
BUCHWALD, WF
.
JOURNAL OF PHARMACEUTICAL SCIENCES,
1984,
73
(02)
:243
-246
[7]
CONTROLLED COMPARISON OF IM MORPHINE AND BUPRENORPHINE FOR ANALGESIA AFTER ABDOMINAL-SURGERY
[J].
COOK, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL FREE HOSP,DEPT SURG,LONDON NW3 2QG,ENGLAND
COOK, PJ
;
JAMES, IM
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL FREE HOSP,DEPT SURG,LONDON NW3 2QG,ENGLAND
JAMES, IM
;
HOBBS, KEF
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL FREE HOSP,DEPT SURG,LONDON NW3 2QG,ENGLAND
HOBBS, KEF
;
BROWNE, DRG
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL FREE HOSP,DEPT SURG,LONDON NW3 2QG,ENGLAND
BROWNE, DRG
.
BRITISH JOURNAL OF ANAESTHESIA,
1982,
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[8]
ANIMAL PHARMACOLOGY OF BUPRENORPHINE, AN ORIPAVINE ANALGESIC AGENT
[J].
COWAN, A
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DEPT PHARMACOL,HULL HU8 7DS,ENGLAND
RECKITT & COLMAN LTD,DEPT PHARMACOL,HULL HU8 7DS,ENGLAND
COWAN, A
;
DOXEY, JC
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DEPT PHARMACOL,HULL HU8 7DS,ENGLAND
RECKITT & COLMAN LTD,DEPT PHARMACOL,HULL HU8 7DS,ENGLAND
DOXEY, JC
;
HARRY, EJR
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DEPT PHARMACOL,HULL HU8 7DS,ENGLAND
RECKITT & COLMAN LTD,DEPT PHARMACOL,HULL HU8 7DS,ENGLAND
HARRY, EJR
.
BRITISH JOURNAL OF PHARMACOLOGY,
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COWEN A, 1977, BRIT J PHARMACOL, V60, P537
[10]
ELECTROCHEMICAL CHROMATOGRAPHIC DETERMINATIONS OF MORPHINE ANTAGONISTS IN BIOLOGICAL-FLUIDS, WITH APPLICATIONS
[J].
DERENDORF, H
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV FLORIDA,J HILLIS MILLER HLTH CTR,COLL PHARM,BEEHIVE,GAINESVILLE,FL 32610
UNIV FLORIDA,J HILLIS MILLER HLTH CTR,COLL PHARM,BEEHIVE,GAINESVILLE,FL 32610
DERENDORF, H
;
ELDIN, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV FLORIDA,J HILLIS MILLER HLTH CTR,COLL PHARM,BEEHIVE,GAINESVILLE,FL 32610
UNIV FLORIDA,J HILLIS MILLER HLTH CTR,COLL PHARM,BEEHIVE,GAINESVILLE,FL 32610
ELDIN, A
;
ELKOUSSI, A
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV FLORIDA,J HILLIS MILLER HLTH CTR,COLL PHARM,BEEHIVE,GAINESVILLE,FL 32610
UNIV FLORIDA,J HILLIS MILLER HLTH CTR,COLL PHARM,BEEHIVE,GAINESVILLE,FL 32610
ELKOUSSI, A
;
GARRETT, ER
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV FLORIDA,J HILLIS MILLER HLTH CTR,COLL PHARM,BEEHIVE,GAINESVILLE,FL 32610
UNIV FLORIDA,J HILLIS MILLER HLTH CTR,COLL PHARM,BEEHIVE,GAINESVILLE,FL 32610
GARRETT, ER
.
JOURNAL OF PHARMACEUTICAL SCIENCES,
1984,
73
(05)
:621
-624
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2
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共 35 条
[1]
THE RADIOIMMUNOASSAY OF BUPRENORPHINE
[J].
BARTLETT, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
BARTLETT, AJ
;
LLOYDJONES, JG
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
LLOYDJONES, JG
;
RANCE, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
RANCE, MJ
;
FLOCKHART, IR
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
FLOCKHART, IR
;
DOCKRAY, GJ
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
DOCKRAY, GJ
;
BENNETT, MRD
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
BENNETT, MRD
;
MOORE, RA
论文数:
0
引用数:
0
h-index:
0
机构:
RECKITT & COLMAN LTD,DIV PHARMACEUT,PHARMACEUT R & D LABS,HULL HU8 7DS,N HUMBERSHIRE,ENGLAND
MOORE, RA
.
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY,
1980,
18
(04)
:339
-345
[2]
SUB-LINGUAL BUPRENORPHINE USED POSTOPERATIVELY - 10-HOUR PLASMA DRUG CONCENTRATION ANALYSIS
[J].
BULLINGHAM, RES
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
BULLINGHAM, RES
;
MCQUAY, HJ
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
MCQUAY, HJ
;
PORTER, EJB
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
PORTER, EJB
;
ALLEN, MC
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
ALLEN, MC
;
MOORE, RA
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
MOORE, RA
.
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY,
1982,
13
(05)
:665
-673
[3]
AN ORAL BUPRENORPHINE AND PARACETAMOL COMBINATION COMPARED WITH PARACETAMOL ALONE - A SINGLE DOSE DOUBLE-BLIND POSTOPERATIVE STUDY
[J].
BULLINGHAM, RES
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
BULLINGHAM, RES
;
MCQUAY, HJ
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
MCQUAY, HJ
;
MOORE, RA
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
MOORE, RA
;
WEIR, L
论文数:
0
引用数:
0
h-index:
0
机构:
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
JOHN RADCLIFFE HOSP,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX3 9DU,ENGLAND
WEIR, L
.
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY,
1981,
12
(06)
:863
-867
[4]
BUPRENORPHINE KINETICS
[J].
BULLINGHAM, RES
论文数:
0
引用数:
0
h-index:
0
机构:
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
BULLINGHAM, RES
;
MCQUAY, HJ
论文数:
0
引用数:
0
h-index:
0
机构:
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
MCQUAY, HJ
;
MOORE, A
论文数:
0
引用数:
0
h-index:
0
机构:
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
MOORE, A
;
BENNETT, MRD
论文数:
0
引用数:
0
h-index:
0
机构:
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
RADCLIFFE INFIRM,NUFFIELD DEPT CLIN BIOCHEM,OXFORD OX2 6HE,ENGLAND
BENNETT, MRD
.
CLINICAL PHARMACOLOGY & THERAPEUTICS,
1980,
28
(05)
:667
-672
[5]
COMPARISON OF BUPRENORPHINE AND PETHIDINE GIVEN INTRAVENOUSLY ON DEMAND TO RELIEVE POST-OPERATIVE PAIN
[J].
CHAKRAVARTY, K
论文数:
0
引用数:
0
h-index:
0
机构:
Jipmer, Pondicherry
CHAKRAVARTY, K
;
TUCKER, W
论文数:
0
引用数:
0
h-index:
0
机构:
Jipmer, Pondicherry
TUCKER, W
;
ROSEN, M
论文数:
0
引用数:
0
h-index:
0
机构:
Jipmer, Pondicherry
ROSEN, M
;
VICKERS, MD
论文数:
0
引用数:
0
h-index:
0
机构:
Jipmer, Pondicherry
VICKERS, MD
.
BRITISH MEDICAL JOURNAL,
1979,
2
(6195)
:895
-897
[6]
STABILITY OF THE "6,14-ENDO-ETHANOTETRAHYDROORIPAVINE ANALGESICS - ACID-CATALYZED REARRANGEMENT OF BUPRENORPHINE
[J].
CONE, EJ
论文数:
0
引用数:
0
h-index:
0
CONE, EJ
;
GORODETZKY, CW
论文数:
0
引用数:
0
h-index:
0
GORODETZKY, CW
;
DARWIN, WD
论文数:
0
引用数:
0
h-index:
0
DARWIN, WD
;
BUCHWALD, WF
论文数:
0
引用数:
0
h-index:
0
BUCHWALD, WF
.
JOURNAL OF PHARMACEUTICAL SCIENCES,
1984,
73
(02)
:243
-246
[7]
CONTROLLED COMPARISON OF IM MORPHINE AND BUPRENORPHINE FOR ANALGESIA AFTER ABDOMINAL-SURGERY
[J].
COOK, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
ROYAL FREE HOSP,DEPT SURG,LONDON NW3 2QG,ENGLAND
COOK, PJ
;
JAMES, IM
论文数:
0
引用数:
0
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