SYNTHESIS OF 7-SUBSTITUTED INDOLES AS POTENTIAL LIGAND PRECURSORS

被引：8

作者：

BLACK, DS ^{[1
]}

DEACON, GB ^{[1
]}

EDWARDS, GL ^{[1
]}

机构：

[1] MONASH UNIV,DEPT CHEM,CLAYTON,VIC 3168,AUSTRALIA

来源：

AUSTRALIAN JOURNAL OF CHEMISTRY | 1991年 / 44卷 / 12期

关键词：

D O I：

10.1071/CH9911771

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Some 7-(pyridin-2'-yl)- and 7-(pyrazol-1'-yl)-indole-2-carboxylic esters (14)-(16) and the related acids (17) and (18) have been synthesized through the Fischer indole cyclizations of the ethyl pyruvate hydrazones (9)-(12), which were in turn derived from the ortho-functionalized anilines (5)-(8) by diazotization and coupling with ethyl 2-methyl-3-oxobutanoate (the Japp-Klingemann reaction).

引用

页码：1771 / 1781

页数：11

共 19 条

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