DESIGN AND SYNTHESIS OF NALTREXONE-DERIVED AFFINITY LABELS WITH NONEQUILIBRIUM OPIOID AGONIST AND ANTAGONIST ACTIVITIES - EVIDENCE FOR THE EXISTENCE OF DIFFERENT MU-RECEPTOR SUBTYPES IN DIFFERENT TISSUES

被引:49
作者
SAYRE, LM
LARSON, DL
TAKEMORI, AE
PORTOGHESE, PS
机构
[1] UNIV MINNESOTA, COLL PHARM, DEPT MED CHEM, MINNEAPOLIS, MN 55455 USA
[2] UNIV MINNESOTA, SCH MED, DEPT PHARMACOL, MINNEAPOLIS, MN 55455 USA
关键词
D O I
10.1021/jm00376a018
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
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页码:1325 / 1335
页数:11
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