PHARMACOLOGICAL ANALYSIS OF BETA-ADRENOCEPTOR-MEDIATED AGONISM IN THE GUINEA-PIG, ISOLATED, RIGHT ATRIUM

被引:20
作者
BLACK, JW
GERSKOWITCH, VP
LEFF, P
SHANKLEY, NP
机构
[1] WELLCOME RES LABS, LANGLEY COURT, BECKENHAM BR3 3BS, KENT, ENGLAND
[2] UNIV LONDON KINGS COLL HOSP, SCH MED, RAYNE INST, LONDON SE5 8RX, ENGLAND
关键词
D O I
10.1111/j.1476-5381.1985.tb16161.x
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:779 / 785
页数:7
相关论文
共 9 条
[1]  
ANGUS JA, 1980, CIRC RES, V65, P1
[2]  
BAKER SP, 1982, J PHARMACOL EXP THER, V220, P247
[3]   OPERATIONAL MODELS OF PHARMACOLOGICAL AGONISM [J].
BLACK, JW ;
LEFF, P .
PROCEEDINGS OF THE ROYAL SOCIETY SERIES B-BIOLOGICAL SCIENCES, 1983, 220 (1219) :141-162
[4]   MECHANISM OF ADENYLATE-CYCLASE ACTIVATION BY CHOLERA TOXIN - INHIBITION OF GTP HYDROLYSIS AT REGULATORY SITE [J].
CASSEL, D ;
SELINGER, Z .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1977, 74 (08) :3307-3311
[5]   MECHANISM OF CHOLERA TOXIN ACTION - COVALENT MODIFICATION OF GUANYL NUCLEOTIDE-BINDING PROTEIN OF ADENYLATE-CYCLASE SYSTEM [J].
CASSEL, D ;
PFEUFFER, T .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1978, 75 (06) :2669-2673
[6]  
DELEAN A, 1980, J BIOL CHEM, V255, P7108
[7]   REGENERATION OF BETA-ADRENERGIC RECEPTORS IN SENESCENT RATS - A STUDY USING AN IRREVERSIBLE BINDING ANTAGONIST [J].
PITHA, J ;
HUGHES, BA ;
KUSIAK, JW ;
DAX, EM ;
BAKER, SP .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1982, 79 (14) :4424-4427
[8]  
RUDOLPH SA, 1977, J BIOL CHEM, V252, P7132
[9]  
VANROSSUM JM, 1963, ARCH INT PHARMACOD T, V143, P240