INTRANASAL ABSORPTION OF A KAPPA-AGONIST ANALGESIC

被引:1
作者
HUSSAIN, MA [1 ]
SCHMIDT, WK [1 ]
BUEHLER, JD [1 ]
机构
[1] DUPONT MERCK PHARMACEUT CO,CNS DIS RES,WILMINGTON,DE 19880
关键词
KAPPA-AGONIST ANALGESIC; NASAL ABSORPTION; BIOAVAILABILITY; PHARMACOKINETICS; ED(50);
D O I
10.1023/A:1018987328143
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
[No abstract available]
引用
收藏
页码:1083 / 1086
页数:4
相关论文
共 15 条
[1]   TRANSNASAL BUTORPHANOL - A NEW METHOD FOR PAIN RELIEF IN POSTCESAREAN SECTION PAIN [J].
ABBOUD, TK ;
ZHU, J ;
GANGOLLY, J ;
LONGHITANO, M ;
SWART, F ;
MAKAR, A ;
CHU, G ;
COOL, M ;
MANTILLA, M ;
KURTZ, N ;
REICH, L .
ACTA ANAESTHESIOLOGICA SCANDINAVICA, 1991, 35 (01) :14-18
[2]  
BLUMBERG H, 1965, P SOC EXP BIOL MED, V118, P763
[3]   CI-977, A NOVEL AND SELECTIVE AGONIST FOR THE KAPPA-OPIOID RECEPTOR [J].
HUNTER, JC ;
LEIGHTON, GE ;
MEECHAM, KG ;
BOYLE, SJ ;
HORWELL, DC ;
REES, DC ;
HUGHES, J .
BRITISH JOURNAL OF PHARMACOLOGY, 1990, 101 (01) :183-189
[4]  
HUSSAIN A, 1979, J PHARM SCI, V68, P196
[5]   INTRANASAL ABSORPTION OF PHYSOSTIGMINE AND ARECOLINE [J].
HUSSAIN, MA ;
MOLLICA, JA .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1991, 80 (08) :750-751
[6]  
JAFFE J H, 1990, P485
[7]  
MARTIN WR, 1976, J PHARMACOL EXP THER, V197, P517
[8]   KAPPA-OPIOID RECEPTORS AND ANALGESIA [J].
MILLAN, MJ .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1990, 11 (02) :70-76
[9]   U-50488H,A PURE KAPPA RECEPTOR AGONIST WITH SPINAL ANALGESIC LOCI IN THE MOUSE [J].
PIERCEY, MF ;
LAHTI, RA ;
SCHROEDER, LA ;
EINSPAHR, FJ ;
BARSUHN, C .
LIFE SCIENCES, 1982, 31 (12-1) :1197-1200
[10]   DUP 747 - SAR STUDY [J].
RAJAGOPALAN, P ;
SCRIBNER, RM ;
PENNEV, P ;
MATTEI, PL ;
KEZAR, HS ;
CHENG, CY ;
CHEESEMAN, RS ;
GANTI, VR ;
JOHNSON, AL ;
WUONOLA, MA ;
SCHMIDT, WK ;
TAM, SW ;
STEINFELS, GF ;
COOK, L .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1992, 2 (07) :721-726