STEREOCONTROLLED SYNTHESIS OF 4,4,4-TRIFLUOROTHREONINE

被引：38

作者：

KITAZUME, T

LIN, JT

YAMAZAKI, T

机构：

[1] Department of Bioengineering, Tokyo Institute of Technology Nagatsuta, Midori-ku, Yokohama

来源：

TETRAHEDRON-ASYMMETRY | 1991年 / 2卷 / 04期

关键词：

D O I：

10.1016/S0957-4166(00)80041-5

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

Stereoisomers of unnatural 4,4,4-trifluorothreonine are obtained through enzymatic resolution, and the absolute configuration of these materials is determined. 4,4,4-Trifluorothreonine thus prepared was evaluated for antifungal or antitumor activity.

引用

页码：235 / 238

页数：4

共 9 条

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