[I-125] IODOBOLPYRAMINE, A HIGHLY SENSITIVE PROBE FOR HISTAMINE H1-RECEPTORS IN GUINEA-PIG BRAIN

被引:37
作者
KORNER, M
BOUTHENET, ML
GANELLIN, CR
GARBARG, M
GROS, C
IFE, RJ
SALES, N
SCHWARTZ, JC
机构
[1] INSERM,CTR PAUL BROCA,UNITE 109 NEUROBIOL,2TER RUE ALESIA,F-75014 PARIS,FRANCE
[2] FAC PHARM PARIS,PHYSIOL LAB,F-75005 PARIS,FRANCE
[3] SK F RES LTD,WELWYN AL6 9AR,HERTS,ENGLAND
关键词
D O I
10.1016/0014-2999(86)90535-2
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:151 / 160
页数:10
相关论文
共 45 条
[1]   AUTO-INHIBITION OF BRAIN HISTAMINE-RELEASE MEDIATED BY A NOVEL CLASS (H-3) OF HISTAMINE-RECEPTOR [J].
ARRANG, JM ;
GARBARG, M ;
SCHWARTZ, JC .
NATURE, 1983, 302 (5911) :832-837
[2]   HISTAMINE SYNTHESIZING AFFERENTS TO HIPPOCAMPAL REGION [J].
BARBIN, G ;
GARBARG, M ;
SCHWARTZ, JC ;
STORMMATHISEN, J .
JOURNAL OF NEUROCHEMISTRY, 1976, 26 (02) :259-263
[3]   HISTAMINE SYNTHESIZING AFFERENTS WITHIN AMYGDALOID COMPLEX AND BED NUCLEUS OF STRIA TERMINALIS OF RAT [J].
BENARI, Y ;
LEGALLASALLE, G ;
BARBIN, G ;
SCHWARTZ, JC ;
GARBARG, M .
BRAIN RESEARCH, 1977, 138 (02) :285-294
[4]   DEFINITION AND ANTAGONISM OF HISTAMINE H2-RECEPTORS [J].
BLACK, JW ;
PARSONS, EM ;
DURANT, CJ ;
DUNCAN, WAM ;
GANELLIN, CR .
NATURE, 1972, 236 (5347) :385-&
[5]   LABELING OF PROTEINS TO HIGH SPECIFIC RADIOACTIVITIES BY CONJUGATION TO A I-125-CONTAINING ACYLATING AGENT - APPLICATION TO RADIOIMMUNOASSAY [J].
BOLTON, AE ;
HUNTER, WM .
BIOCHEMICAL JOURNAL, 1973, 133 (03) :529-538
[6]   CIMETIDINE - NON-THIOUREA H2-RECEPTOR ANTAGONIST [J].
BRIMBLECOMBE, RW ;
DUNCAN, WAM ;
DURANT, GJ ;
EMMETT, JC ;
GANELLIN, CR ;
PARSONS, ME .
JOURNAL OF INTERNATIONAL MEDICAL RESEARCH, 1975, 3 (02) :86-92
[7]   A RAPID FILTRATION ASSAY FOR SOLUBLE RECEPTORS USING POLYETHYLENIMINE-TREATED FILTERS [J].
BRUNS, RF ;
LAWSONWENDLING, K ;
PUGSLEY, TA .
ANALYTICAL BIOCHEMISTRY, 1983, 132 (01) :74-81
[8]   HETEROGENEITY OF HISTAMINE H1-RECEPTORS - SPECIES VARIATIONS IN [MEPYRAMINE-H-3 BINDING OF BRAIN MEMBRANES [J].
CHANG, RSL ;
TRAN, VT ;
SNYDER, SH .
JOURNAL OF NEUROCHEMISTRY, 1979, 32 (06) :1653-1663
[9]   HISTAMINE H1-RECEPTORS IN BRAIN LABELED WITH MEPYRAMINE-H-3 [J].
CHANG, RSL ;
TRAN, VT ;
SNYDER, SH .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1978, 48 (04) :463-464
[10]   HISTAMINE STIMULATION OF INOSITOL 1-PHOSPHATE ACCUMULATION IN LITHIUM-TREATED SLICES FROM REGIONS OF GUINEA-PIG BRAIN [J].
DAUM, PR ;
DOWNES, CP ;
YOUNG, JM .
JOURNAL OF NEUROCHEMISTRY, 1984, 43 (01) :25-32