EFFICIENT AND SELECTIVE METHOD FOR SYNTHESIS OF 2-(4-FLUOROPHENYL)-1-(2-HYDROXYETHYL)-5-NITROIMIDAZOLE (FLUNIDAZOLE)

被引：8

作者：

GRABOWSK.EJ ^{[1
]}

LIU, TMH ^{[1
]}

SALCE, L ^{[1
]}

SCHOENEW.EF ^{[1
]}

机构：

[1] MERCK SHARP & DOHME,RES LABS,RAHWAY,NJ 07065

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1974年 / 17卷 / 05期

关键词：

D O I：

10.1021/jm00251a020

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：547 / 549

页数：3

共 18 条

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GRIMISON, A ;

RIDD, JH ;

SMITH, BV .

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[4] THE MECHANISMS OF N-SUBSTITUTION IN GLYOXALINE DERIVATIVES .1. INTRODUCTION, AND STUDY OF PROTOTROPIC EQUILIBRIA INVOLVING 4(5)-NITROGLYOXALINE [J].

GRIMISON, A ;

RIDD, JH ;

SMITH, BV .

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[5]

Hofmann K., 1953, IMIDAZOLE ITS DERIVA

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[7] TREATMENT OF UROGENITAL TRICHOMONIASIS [J].

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AMERICAN JOURNAL OF OBSTETRICS AND GYNECOLOGY, 1973, 115 (04) :587-588

[8]

KOLLONITSCH J, 1969, Patent No. 3471512

[9]

KOLLONITSCH J, 1969, Patent No. 3471511

[10]

KOLLONITSCH J, 1971, Patent No. 42923

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