STEREOSELECTIVE SYNTHESES OF PEPTIDE DERIVATIVES WITH 2-ACETAMIDO-3,4,6-TRI-O-ACETYL-1-AMINO-2-DEOXY-BETA-D-GLUCOPYRANOSE BY 4-COMPONENT CONDENSATION

被引：54

作者：

LEHNHOFF, S ^{[1
]}

GOEBEL, M ^{[1
]}

KARL, RM ^{[1
]}

KLOSEL, R ^{[1
]}

UGI, I ^{[1
]}

机构：

[1] TECH UNIV MUNICH,INST ORGAN CHEM & BIOCHEM,D-85747 GARCHING,GERMANY

来源：

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH | 1995年 / 34卷 / 10期

关键词：

ASYMMETRIC SYNTHESES; CHIRAL AUXILIARIES; PEPTIDE SYNTHESES; 4-COMPONENT REACTIONS;

D O I：

10.1002/anie.199511041

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Diastereoisomeric excesses greater than 99% are obtained for the majority of the stereoselective four‐component condensations (a), if the amino glucopyranose 1 is used as the sugar component Y‐NH2. (Figure Presented.) Copyright © 1995 by VCH Verlagsgesellschaft mbH, Germany

引用

页码：1104 / 1107

页数：4

共 40 条

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