HIV-1 PROTEASE INHIBITORS - DEVELOPMENT, STATUS, AND POTENTIAL ROLE IN THE TREATMENT OF AIDS

被引:22
作者
LANG, M
ROESEL, J
机构
关键词
D O I
10.1002/ardp.19933261202
中图分类号
R914 [药物化学];
学科分类号
100701 ;
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页码:921 / 924
页数:4
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共 58 条
[1]   CGP-53437, AN ORALLY BIOAVAILABLE INHIBITOR OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 PROTEASE WITH POTENT ANTIVIRAL ACTIVITY [J].
ALTERI, E ;
BOLD, G ;
COZENS, R ;
FAESSLER, A ;
KLIMKAIT, T ;
LANG, M ;
LAZDINS, J ;
PONCIONI, B ;
ROESEL, JL ;
SCHNEIDER, P ;
WALKER, M ;
WOODSCOOK, K .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1993, 37 (10) :2087-2092
[2]   ISOLATION OF A T-LYMPHOTROPIC RETROVIRUS FROM A PATIENT AT RISK FOR ACQUIRED IMMUNE-DEFICIENCY SYNDROME (AIDS) [J].
BARRESINOUSSI, F ;
CHERMANN, JC ;
REY, F ;
NUGEYRE, MT ;
CHAMARET, S ;
GRUEST, J ;
DAUGUET, C ;
AXLERBLIN, C ;
VEZINETBRUN, F ;
ROUZIOUX, C ;
ROZENBAUM, W ;
MONTAGNIER, L .
SCIENCE, 1983, 220 (4599) :868-871
[3]  
BILLICH S, 1988, J BIOL CHEM, V263, P17905
[4]   SYNTHETIC NON-PEPTIDE INHIBITORS OF HIV PROTEASE [J].
BLUMENSTEIN, JJ ;
COPELAND, TD ;
OROSZLAN, S ;
MICHEJDA, CJ .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1989, 163 (02) :980-987
[5]   FLAVONES ARE INHIBITORS OF HIV-1 PROTEINASE [J].
BRINKWORTH, RI ;
STOERMER, MJ ;
FAIRLIE, DP .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1992, 188 (02) :631-637
[6]   MICROBIAL TRANSFORMATION OF L-696,474, A NOVEL CYTOCHALASIN AS AN INHIBITOR OF HIV-1 PROTEASE [J].
CHEN, TS ;
DOSS, GA ;
HSU, A ;
HSU, A ;
LINGHAM, RB ;
WHITE, RF ;
MONAGHAN, RL .
JOURNAL OF NATURAL PRODUCTS, 1993, 56 (05) :755-761
[7]   HIV-1 PROTEASE SPECIFICITY OF PEPTIDE CLEAVAGE IS SUFFICIENT FOR PROCESSING OF GAG AND POL POLYPROTEINS [J].
DARKE, PL ;
NUTT, RF ;
BRADY, SF ;
GARSKY, VM ;
CICCARONE, TM ;
LEU, CT ;
LUMMA, PK ;
FREIDINGER, RM ;
VEBER, DF ;
SIGAL, IS .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1988, 156 (01) :297-303
[8]   HUMAN-IMMUNODEFICIENCY-VIRUS PROTEASE - A TARGET FOR AIDS THERAPY [J].
DEBOUCK, C ;
METCALF, BW .
DRUG DEVELOPMENT RESEARCH, 1990, 21 (01) :1-17
[9]   THE HIV-1 PROTEASE AS A THERAPEUTIC TARGET FOR AIDS [J].
DEBOUCK, C .
AIDS RESEARCH AND HUMAN RETROVIRUSES, 1992, 8 (02) :153-164
[10]  
DELFRAISSY JF, 1993, 9TH INT C AIDS BERL