SELECTIVE INDUCTION AND INHIBITION OF THE COMPONENTS OF 7-ETHOXYCOUMARIN O-DEETHYLASE ACTIVITY IN THE RAT

被引:23
作者
BOOBIS, AR
WHYTE, C
DAVIES, DS
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关键词
D O I
10.3109/00498258609043526
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:233 / 238
页数:6
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共 19 条
[1]   METABOLISM OF 2-ACETYLAMINOFLUORENE BY 8 DIFFERENT FORMS OF CYTOCHROME-P-450 ISOLATED FROM RAT-LIVER [J].
ASTROM, A ;
DEPIERRE, JW .
CARCINOGENESIS, 1985, 6 (01) :113-120
[2]   MONO-OXYGENASE ACTIVITY OF HUMAN-LIVER IN MICROSOMAL FRACTIONS OF NEEDLE-BIOPSY SPECIMENS [J].
BOOBIS, AR ;
BRODIE, MJ ;
KAHN, GC ;
FLETCHER, DR ;
SAUNDERS, JH ;
DAVIES, DS .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1980, 9 (01) :11-19
[3]   BIPHASIC O-DEETHYLATION OF PHENACETIN AND 7-ETHOXYCOUMARIN BY HUMAN AND RAT-LIVER MICROSOMAL FRACTIONS [J].
BOOBIS, AR ;
KAHN, GC ;
WHYTE, C ;
BRODIE, MJ ;
DAVIES, DS .
BIOCHEMICAL PHARMACOLOGY, 1981, 30 (17) :2451-2456
[4]  
GREENLEE WF, 1978, J PHARMACOL EXP THER, V205, P596
[5]   PURIFICATION AND CHARACTERIZATION OF MICROSOMAL CYTOCHROME-P-450S [J].
GUENGERICH, FP ;
DANNAN, GA ;
WRIGHT, ST ;
MARTIN, MV ;
KAMINSKY, LS .
XENOBIOTICA, 1982, 12 (11) :701-716
[6]  
GUENGERICH FP, 1977, J BIOL CHEM, V252, P3970
[7]  
GUENGERICH FP, 1978, J BIOL CHEM, V253, P7931
[8]  
JOHNSON EF, 1979, MOL PHARMACOL, V15, P708
[9]   METABOLIC PROCESSING OF 2-ACETYLAMINOFLUORENE BY MICROSOMES AND 6 HIGHLY PURIFIED CYTOCHROME-P-450 FORMS FROM RABBIT LIVER [J].
MCMANUS, ME ;
MINCHIN, RF ;
SANDERSON, N ;
SCHWARTZ, D ;
JOHNSON, EF ;
THORGEIRSSON, SS .
CARCINOGENESIS, 1984, 5 (12) :1717-1723
[10]  
MITCHELL JR, 1973, DRUG METAB DISPOS, V1, P418