RECENT PROGRESS IN THE MEDICINAL CHEMISTRY OF 2,4-DIAMINOPYRIMIDINES

被引:85
作者
ROTH, B [1 ]
CHENG, CC [1 ]
机构
[1] UNIV KANSAS, MED CTR, MED CTR, MID AMER CANC CTR, KANSAS CITY, KS 66103 USA
关键词
D O I
10.1016/S0079-6468(08)70332-1
中图分类号
学科分类号
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页码:269 / 331
页数:63
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共 411 条
[1]  
ALBERTO P, 1978, CANCER CHEMOTH PHARM, V1, P101
[2]  
ALBRECHT AM, 1970, MOL PHARMACOL, V6, P323
[3]   THE HALOGENATION OF 4-AMINO-4-DEOXY-N-10-METHYLPTEROYLGLUTAMIC ACID (METHOTREXATE) AND OTHER PTEROYLGLUTAMIC ACID DERIVATIVES [J].
ANGIER, RB ;
CURRAN, WV .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1959, 81 (11) :2814-2818
[4]   THE STRUCTURE AND SYNTHESIS OF THE LIVER L-CASEI FACTOR [J].
ANGIER, RB ;
BOOTHE, JH ;
HUTCHINGS, BL ;
MOWAT, JH ;
SEMB, J ;
STOKSTAD, ELR ;
SUBBAROW, Y ;
WALLER, CW ;
COSULICH, DB ;
FAHRENBACH, MJ ;
HULTQUIST, ME ;
KUH, E ;
NORTHEY, EH ;
SEEGER, DR ;
SICKELS, JP ;
SMITH, JM .
SCIENCE, 1946, 103 (2683) :667-669
[5]   QUINAZOLINES AS INHIBITORS OF DIHYDROFOLATE REDUCTASE .1. [J].
ASHTON, WT ;
WALKER, FC ;
HYNES, JB .
JOURNAL OF MEDICINAL CHEMISTRY, 1973, 16 (06) :694-697
[6]  
AYUSAWA D, 1981, CANCER RES, V41, P1497
[7]  
BACCANARI DP, 1981, J BIOL CHEM, V256, P1738
[8]   DIHYDROFOLATE-REDUCTASE HYSTERESIS AND ITS EFFECT ON INHIBITOR BINDING ANALYSES [J].
BACCANARI, DP ;
JOYNER, SS .
BIOCHEMISTRY, 1981, 20 (07) :1710-1716
[9]  
BACCANARI DP, 1981, FED PROC, V40, P1748
[10]  
BAKER BJ, 1981, 12TH GEN ASS INT UN