SGD 101-75 IS DISTINGUISHED FROM OTHER SELECTIVE ALPHA-1-ADRENOCEPTOR AGONISTS BY THE INHIBITION OF ITS PRESSOR-RESPONSES BY CALCIUM ENTRY BLOCKADE AND VASODILATATION IN PITHED RATS AND CATS

被引:59
作者
TIMMERMANS, PBMWM
THOOLEN, MJMC
MATHY, MJ
WILFFERT, B
DEJONGE, A
VANZWIETEN, PA
机构
关键词
D O I
10.1016/0014-2999(83)90307-2
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:187 / 192
页数:6
相关论文
共 22 条
[1]  
CAMBRIDGE D, 1977, BRIT J PHARMACOL, V59, P514
[2]  
CHADWICK MA, 1983, BR J PHARM, V78, pP155
[3]   OCCURRENCE OF ALPHA-1S-ADRENOCEPTORS IN THE MOUSE BUT NOT IN THE RABBIT ISOLATED ANOCOCCYGEUS PREPARATIONS [J].
COATES, J ;
WEETMAN, DF .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 78 (01) :117-122
[4]   THE EXISTENCE OF A NEW SUBTYPE OF ALPHA-ADRENOCEPTOR ON THE RAT ANOCOCCYGEUS IS REVEALED BY SGD 101/75 AND PHENOXYBENZAMINE [J].
COATES, J ;
JAHN, U ;
WEETMAN, DF .
BRITISH JOURNAL OF PHARMACOLOGY, 1982, 75 (03) :549-552
[5]   CAPTOPRIL IMPAIRS THE VASCULAR SMOOTH-MUSCLE CONTRACTION MEDIATED BY POSTSYNAPTIC ALPHA-2-ADRENOCEPTORS IN THE PITHED RAT [J].
DEJONGE, A ;
WILFFERT, B ;
KALKMAN, HO ;
VANMEEL, JCA ;
THOOLEN, MJMC ;
TIMMERMANS, PBMWM ;
VANZWIETEN, PA .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1981, 74 (04) :385-386
[6]   A LIPOPHILIC, SELECTIVE ALPHA-1-ADRENOCEPTOR AGONIST - 2-(2-CHLORO-5-TRIFLUOROMETHYLPHENYLIMINO) IMIDAZOLIDINE (ST 587) [J].
DEJONGE, A ;
VANMEEL, JCA ;
TIMMERMANS, PBMWM ;
VANZWIETEN, PA .
LIFE SCIENCES, 1981, 28 (18) :2009-2016
[7]   EFFECT OF CONVERTING ENZYME-INHIBITION AND ANGIOTENSIN RECEPTOR BLOCKADE ON THE VASOCONSTRICTION MEDIATED BY ALPHA-1-ADRENOCEPTOR AND ALPHA-2-ADRENOCEPTOR STIMULATION IN PITHED NORMOTENSIVE RATS [J].
DEJONGE, A ;
KNAPE, JTA ;
VANMEEL, JCA ;
KALKMAN, HO ;
WILFFERT, B ;
THOOLEN, MJMC ;
TIMMERMANNS, PBMWM ;
VANZWIETEN, PA .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 321 (04) :309-313
[8]  
GIBSON A, 1983, BR J PHARM, V3, P1
[9]   A METHOD OF STIMULATING DIFFERENT SEGMENTS OF AUTONOMIC OUTFLOW FROM SPINAL COLUMN TO VARIOUS ORGANS IN PITHED CAT AND RAT [J].
GILLESPIE, JS ;
MACLAREN, A ;
POLLOCK, D .
BRITISH JOURNAL OF PHARMACOLOGY, 1970, 40 (02) :257-+
[10]   DIFFERENTIAL INTERACTIONS OF CLONIDINE AND METHOXAMINE WITH THE POSTSYNAPTIC ALPHA-ADRENOCEPTOR OF RABBIT MAIN PULMONARY-ARTERY [J].
HOLCK, MI ;
JONES, CHM ;
HAEUSLER, G .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1983, 5 (02) :240-248