SPECIFIC HIV-1 REVERSE-TRANSCRIPTASE INHIBITORS

被引:16
作者
DEBYSER, Z
PAUWELS, R
ANDRIES, K
DE CLERCQ, E
机构
[1] CATHOLIC UNIV LEUVEN, REGA INST MED RES, B-3000 LOUVAIN, BELGIUM
[2] JANSSEN RES FDN, B-2340 BEERSE, BELGIUM
来源
JOURNAL OF ENZYME INHIBITION | 1992年 / 6卷 / 01期
关键词
HIV-1; REVERSE TRANSCRIPTASE; INHIBITORS; AZT; HEPT; TIBO;
D O I
10.3109/14756369209041355
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
[No abstract available]
引用
收藏
页码:47 / 53
页数:7
相关论文
共 17 条
  • [1] ARNOLD E, 1991, ADV VIRUS RES, V39, P1
  • [2] BABA M, 1991, MOL PHARMACOL, V39, P805
  • [3] POTENT AND SELECTIVE-INHIBITION OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 (HIV-1) BY 5-ETHYL-6-PHENYLTHIOURACIL DERIVATIVES THROUGH THEIR INTERACTION WITH THE HIV-1 REVERSE-TRANSCRIPTASE
    BABA, M
    DECLERCQ, E
    TANAKA, H
    UBASAWA, M
    TAKASHIMA, H
    SEKIYA, K
    NITTA, I
    UMEZU, K
    NAKASHIMA, H
    MORI, S
    SHIGETA, S
    WALKER, RT
    MIYASAKA, T
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1991, 88 (06) : 2356 - 2360
  • [4] HIGHLY SPECIFIC-INHIBITION OF HUMAN IMMUNODEFICIENCY VIRUS TYPE-1 BY A NOVEL 6-SUBSTITUTED ACYCLOURIDINE DERIVATIVE
    BABA, M
    TANAKA, H
    DECLERCQ, E
    PAUWELS, R
    BALZARINI, J
    SCHOLS, D
    NAKASHIMA, H
    PERNO, CF
    WALKER, RT
    MIYASAKA, T
    [J]. BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1989, 165 (03) : 1375 - 1381
  • [5] AN ANTIVIRAL TARGET ON REVERSE-TRANSCRIPTASE OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 REVEALED BY TETRAHYDROIMIDAZO[4,5,1-JK][1,4]BENZODIAZEPIN-2(1H)-ONE AND TETRAHYDROIMIDAZO-[4,5,1-JK][1,4]BENZODIAZEPIN-2(1H)-ONE-THIONE DERIVATIVES
    DEBYSER, Z
    PAUWELS, R
    ANDRIES, K
    DESMYTER, J
    KUKLA, M
    JANSSEN, PAJ
    DECLERCQ, E
    [J]. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1991, 88 (04) : 1451 - 1455
  • [6] DECLERCQ E, 1991, J ACQ IMMUN DEF SYND, V4, P207
  • [7] NEW ACQUISITIONS IN THE DEVELOPMENT OF ANTI-HIV AGENTS
    DECLERCQ, E
    [J]. ANTIVIRAL RESEARCH, 1989, 12 (01) : 1 - 19
  • [8] FURFINE ES, 1991, J BIOL CHEM, V266, P406
  • [9] GOLDMAN ME, 1991, 7 INT C AIDS FLOR
  • [10] GENOME ORGANIZATION AND TRANSACTIVATION OF THE HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-2
    GUYADER, M
    EMERMAN, M
    SONIGO, P
    CLAVEL, F
    MONTAGNIER, L
    ALIZON, M
    [J]. NATURE, 1987, 326 (6114) : 662 - 669