MECHANISM OF INACTIVATION OF THYROID PEROXIDASE BY THIOUREYLENE DRUGS

被引:94
作者
ENGLER, H [1 ]
TAUROG, A [1 ]
NAKASHIMA, T [1 ]
机构
[1] UNIV TEXAS,HLTH SCI CTR,DEPT PHARMACOL,DALLAS,TX 75235
关键词
D O I
10.1016/0006-2952(82)90296-9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:3801 / 3806
页数:6
相关论文
共 20 条
[2]   THIOUREA AND CYANAMIDE AS INHIBITORS OF THYROID PEROXIDASE - ROLE OF IODIDE [J].
DAVIDSON, B ;
SOODAK, M ;
STROUT, HV ;
NEARY, JT ;
NAKAMURA, C ;
MALOOF, F .
ENDOCRINOLOGY, 1979, 104 (04) :919-924
[3]   IRREVERSIBLE INACTIVATION OF THYROID PEROXIDASE BY METHYLMERCAPTOIMIDAZOLE, THIOURACIL, AND PROPYLTHIOURACIL INVITRO AND ITS RELATIONSHIP TO INVIVO FINDINGS [J].
DAVIDSON, B ;
SOODAK, M ;
NEARY, JT ;
STROUT, HV ;
KIEFFER, JD ;
MOVER, H ;
MALOOF, F .
ENDOCRINOLOGY, 1978, 103 (03) :871-882
[4]  
EDELHOCH H, 1979, J BIOL CHEM, V254, P822
[7]  
MALOOF F, 1965, CURRENT TOPICS THYRO, P277
[8]  
MICHOT JL, 1979, J BIOL CHEM, V254, P2205
[9]  
MORRIS DR, 1966, J BIOL CHEM, V241, P3582
[10]   MECHANISM OF ACTION OF THIOUREYLENE ANTI-THYROID DRUGS - FACTORS AFFECTING INTRATHYROIDAL METABOLISM OF PROPYLTHIOURACIL AND METHIMAZOLE IN RATS [J].
NAKASHIMA, T ;
TAUROG, A ;
RIESCO, G .
ENDOCRINOLOGY, 1978, 103 (06) :2187-2197