ANALOGS OF 1,3-DIPROPYL-8-PHENYLXANTHINE - ENHANCEMENT OF SELECTIVITY AT ADENOSINE-A1-RECEPTORS BY ARYL SUBSTITUENTS

被引：35

作者：

DALY, JW

PADGETT, WL

SHAMIM, MT

机构：

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1986年 / 29卷 / 08期

关键词：

D O I：

10.1021/jm00158a034

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1520 / 1524

页数：5

共 26 条

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[5] EVIDENCE THAT THE P1-PURINOCEPTOR IN THE GUINEA-PIG TAENIA-COLI IS AN A2-SUBTYPE [J].

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[7] EFFECTS OF AN ADENOSINE-RECEPTOR ANTAGONIST ON INSULIN-RESISTANCE IN SOLEUS MUSCLE FROM OBESE ZUCKER RATS [J].

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[8] ANTAGONISM OF PRESYNAPTIC ADENOSINE RECEPTORS BY THEOPHYLLINE 9-BETA-D-RIBOSIDE AND 8-PHENYLTHEOPHYLLINE [J].

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[9] COMPARISON OF THE POTENCY OF 8-PHENYLTHEOPHYLLINE AS AN ANTAGONIST AT A1 AND A2 ADENOSINE RECEPTORS IN ATRIA AND AORTA FROM THE GUINEA-PIG [J].

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[10] 8-PHENYLTHEOPHYLLINE POTENTIATES THE ELECTRICAL-ACTIVITY EVOKED IN HIPPOCAMPAL SLICES [J].

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