EVALUATION OF POTENTIAL CAUSES FOR THE INCOMPLETE BIOAVAILABILITY OF FUROSEMIDE - GASTRIC 1ST-PASS METABOLISM

被引:184
作者
LEE, MG [1 ]
CHIOU, WL [1 ]
机构
[1] UNIV ILLINOIS,COLL PHARM,DEPT PHARMACODYNAM,CHICAGO,IL 60612
来源
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS | 1983年 / 11卷 / 06期
关键词
D O I
10.1007/BF01059061
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:623 / 640
页数:18
相关论文
共 45 条
[1]   DISTRIBUTION, ELIMINATION AND NATRIURETIC EFFECT OF FUROSEMIDE IN PATIENTS WITH SEVERE ARTERIAL-HYPERTENSION [J].
ANDREASEN, F ;
PEDERSEN, OL ;
MIKKELSEN, E .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1978, 14 (04) :237-244
[2]   INVITRO STUDIES ON THE HYDROLYSIS OF FRUSEMIDE IN GASTROINTESTINAL JUICES [J].
ANDREASEN, F ;
BOTKER, HE ;
LORENTZEN, K .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1982, 14 (02) :306-309
[3]  
BAKER HJ, 1979, LABORATORY RAT, V1, P87
[4]   FATE OF FUROSEMIDE IN MAN [J].
BEERMANN, B ;
DALEN, E ;
LINDSTROM, B ;
ROSEN, A .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1975, 9 (01) :57-61
[5]   PHARMACOKINETICS-PHARMACODYNAMICS OF FUROSEMIDE IN MAN - REVIEW [J].
BENET, LZ .
JOURNAL OF PHARMACOKINETICS AND BIOPHARMACEUTICS, 1979, 7 (01) :1-27
[6]   DETERMINANTS OF RESPONSE TO FRUSEMIDE IN NORMAL SUBJECTS [J].
BRANCH, RA ;
ROBERTS, CJC ;
HOMEIDA, M ;
LEVINE, D .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1977, 4 (02) :121-127
[7]   ABSORPTION AND DISPOSITION OF FUROSEMIDE IN CONGESTIVE HEART-FAILURE [J].
BRATER, DC ;
SEIWELL, R ;
ANDERSON, S ;
BURDETTE, A ;
DEHMER, GJ ;
CHENNAVASIN, P .
KIDNEY INTERNATIONAL, 1982, 22 (02) :171-176
[8]   PHARMACOKINETICS OF DRUGS IN BLOOD III - METABOLISM OF PROCAINAMIDE AND STORAGE EFFECT OF BLOOD-SAMPLES [J].
CHEN, ML ;
LEE, MG ;
CHIOU, WL .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1983, 72 (05) :572-574
[9]   ARTERIAL AND VENOUS-BLOOD SAMPLING IN PHARMACOKINETIC STUDIES - GRISEOFULVIN [J].
CHEN, ML ;
LAM, G ;
LEE, MG ;
CHIOU, WL .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1982, 71 (12) :1386-1389
[10]   PLASMA AREA METHOD IN RELATIVE BIOAVAILABILITY EVALUATION OF DRUGS WITH CHANGING BIOLOGICAL HALF-LIVES [J].
CHIOU, WL ;
LUI, CY ;
LAM, G .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1981, 70 (01) :109-112