IN-VITRO BUT NOT IN-VIVO INHIBITION OF CYP2D6 BY PHENETHYL ISOTHIOCYANATE (PEITC), A CONSTITUENT OF WATERCRESS

被引:14
作者
CAPORASO, N
WHITEHOUSE, J
MONKMAN, S
BOUSTEAD, C
ISSAQ, H
FOX, S
MORSE, MA
IDLE, JR
CHUNG, FL
机构
[1] AMER HLTH FDN,VALHALLA,NY 10595
[2] UNIV NEWCASTLE UPON TYNE,NEWCASTLE TYNE NE1 7RU,TYNE & WEAR,ENGLAND
[3] NCI,FREDERICK CANC RES & DEV CTR,PROGRAM RESOURCES INC DYNCORP,CHEM SYNTH & ANAL LAB,FREDERICK,MD 21702
来源
PHARMACOGENETICS | 1994年 / 4卷 / 05期
关键词
D O I
10.1097/00008571-199410000-00006
中图分类号
Q81 [生物工程学(生物技术)]; Q93 [微生物学];
学科分类号
071005 ; 0836 ; 090102 ; 100705 ;
摘要
[No abstract available]
引用
收藏
页码:275 / 280
页数:6
相关论文
共 40 条
[1]   DEBRISOQUIN OXIDATION GENOTYPE AND SUSCEPTIBILITY TO LUNG-CANCER [J].
AGUNDEZ, JAG ;
MARTINEZ, C ;
LADERO, JM ;
LEDESMA, MC ;
RAMOS, JM ;
MARTIN, R ;
RODRIGUEZ, A ;
JARA, C ;
BENITEZ, J .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1994, 55 (01) :10-14
[2]   HYDROXYLATION POLYMORPHISMS OF DEBRISOQUINE AND MEPHENYTOIN IN EUROPEAN POPULATIONS [J].
ALVAN, G ;
BECHTEL, P ;
ISELIUS, L ;
GUNDERTREMY, U .
EUROPEAN JOURNAL OF CLINICAL PHARMACOLOGY, 1990, 39 (06) :533-537
[3]  
AYESH R, 1984, NATURE, V312, P1669
[4]   POLYMORPHIC OXIDATION OF DEBRISOQUINE IN BLADDER-CANCER [J].
BENITEZ, J ;
LADERO, JM ;
FERNANDEZGUNDIN, MJ ;
LLERENA, A ;
COBALEDA, J ;
MARTINEZ, C ;
MUNOZ, JJ ;
VARGAS, E ;
PRADOS, J ;
GONZALEZROZAS, F ;
RODRIGUEZMOLINA, J ;
USON, AC .
ANNALS OF MEDICINE, 1990, 22 (03) :157-160
[5]   EXTENSIVE METABOLIZERS OF DEBRISOQUINE BECOME POOR METABOLIZERS DURING QUINIDINE TREATMENT [J].
BROSEN, K ;
GRAM, LF ;
HAGHFELT, T ;
BERTILSSON, L .
PHARMACOLOGY & TOXICOLOGY, 1987, 60 (04) :312-314
[6]   THE DISTRIBUTION OF DEBRISOQUINE METABOLIC PHENOTYPES AND IMPLICATIONS FOR THE SUGGESTED ASSOCIATION WITH LUNG-CANCER RISK [J].
CAPORASO, N ;
PICKLE, LW ;
BALE, S ;
AYESH, R ;
HETZEL, M ;
IDLE, J .
GENETIC EPIDEMIOLOGY, 1989, 6 (04) :517-524
[7]  
CAPORASO N, 1991, ARCH INTERN MED, V191, P1985
[8]  
CAPORASO N, 1992, P AM ASSOC CANC RES, V33, P1733
[9]   LUNG-CANCER AND THE DEBRISOQUINE METABOLIC PHENOTYPE [J].
CAPORASO, NE ;
TUCKER, MA ;
HOOVER, RN ;
HAYES, RB ;
PICKLE, LW ;
ISSAQ, HJ ;
MUSCHIK, GM ;
GREENGALLO, L ;
BUIVYS, D ;
AISNER, S ;
RESAU, JH ;
TRUMP, BF ;
TOLLERUD, D ;
WESTON, A ;
HARRIS, CC .
JOURNAL OF THE NATIONAL CANCER INSTITUTE, 1990, 82 (15) :1264-1272
[10]   GENETICALLY-DETERMINED DEBRISOQUINE OXIDATION CAPACITY IN BLADDER-CANCER [J].
CARTWRIGHT, RA ;
PHILIP, PA ;
ROGERS, HJ ;
GLASHAN, RW .
CARCINOGENESIS, 1984, 5 (09) :1191-1192