RENIN INHIBITORS - DESIGN AND SYNTHESIS OF A NEW CLASS OF CONFORMATIONALLY RESTRICTED ANALOGS OF ANGIOTENSINOGEN

被引：49

作者：

SHAM, HL

BOLIS, G

STEIN, HH

FESIK, SW

MARCOTTE, PA

PLATTNER, JJ

REMPEL, CA

GREER, J

机构：

来源：

关键词：

D O I：

10.1021/jm00397a003

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：284 / 295

页数：12

共 52 条

[1] 3-DIMENSIONAL STRUCTURE OF HUMAN RENIN
AKAHANE, K
UMEYAMA, H
NAKAGAWA, S
MORIGUCHI, I
HIROSE, S
IIZUKA, K
MURAKAMI, K
[J]. HYPERTENSION, 1985, 7 (01) : 3 - 12
[2] ANDREEVA NS, 1984, J BIOL CHEM, V259, P1353
[3] [Anonymous], 1965, ORG SYNTH
[4] BANGHAM DR, 1975, CLIN SCI MOL MED, V48, pS135
[5] PROTEIN DATA BANK - COMPUTER-BASED ARCHIVAL FILE FOR MACROMOLECULAR STRUCTURES
BERNSTEIN, FC
KOETZLE, TF
WILLIAMS, GJB
MEYER, EF
BRICE, MD
RODGERS, JR
KENNARD, O
SHIMANOUCHI, T
TASUMI, M
[J]. JOURNAL OF MOLECULAR BIOLOGY, 1977, 112 (03) : 535 - 542
[6] 3-DIMENSIONAL STRUCTURE, SPECIFICITY AND CATALYTIC MECHANISM OF RENIN
BLUNDELL, T
SIBANDA, BL
PEARL, L
[J]. NATURE, 1983, 304 (5923) : 273 - 275
[7] BOGER J, 1985, ANNU REP MED CHEM, V20, P257
[8] RENIN INHIBITORS - SYNTHESES OF SUBNANOMOLAR, COMPETITIVE, TRANSITION-STATE ANALOG INHIBITORS CONTAINING A NOVEL ANALOG OF STATINE
BOGER, J
PAYNE, LS
PERLOW, DS
LOHR, NS
POE, M
BLAINE, EH
ULM, EH
SCHORN, TW
LAMONT, BI
LIN, TY
KAWAI, M
RICH, DH
VEBER, DF
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1985, 28 (12) : 1779 - 1790
[9] BOGER J, 1983, PEPTIDES STRUCTURE F, P569
[10] NEW METHOD FOR METHYLATION OF AMINES
BORCH, RF
HASSID, AI
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1972, 37 (10) : 1673 - &