INVIVO BINDING OF SPIROPERIDOL AND BROMOSPIROPERIDOL AT LOW DRUG LOADINGS

被引:6
作者
DEJESUS, OT
REVENAUGH, JR
DINERSTEIN, RJ
FRIEDMAN, AM
机构
[1] UNIV CHICAGO,DEPT PHARMACOL & PHYSIOL SCI,CHICAGO,IL 60637
[2] ARGONNE NATL LAB,ARGONNE,IL 60439
关键词
D O I
10.1016/0024-3205(84)90517-4
中图分类号
R-3 [医学研究方法]; R3 [基础医学];
学科分类号
1001 ;
摘要
引用
收藏
页码:2165 / 2168
页数:4
相关论文
共 19 条
[1]  
BERGER G, 1981, J LABELLED COMPD RAD, V18, P5
[2]  
Clark AJ., 1933, MODE ACTION DRUGS CE
[3]   PREPARATION AND PURIFICATION OF BR-77-LABELED PARA-BROMOSPIROPERIDOL SUITABLE FOR INVIVO DOPAMINE RECEPTOR STUDIES [J].
DEJESUS, OT ;
FRIEDMAN, AM ;
PRASAD, A ;
REVENAUGH, JR .
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 1983, 20 (06) :745-756
[4]  
DUELFER T, 1982, J NUCL MED, V23, pP13
[5]  
ECKELMAN WC, 1979, J NUCL MED, V20, P350
[6]   BIOCHEMICAL DEMONSTRATION OF DOPAMINERGIC RECEPTORS IN RAT AND HUMAN-BRAIN USING (H-3)SPIROPERIDOL [J].
FIELDS, JZ ;
REISINE, TD ;
YAMAMURA, HI .
BRAIN RESEARCH, 1977, 136 (03) :578-584
[7]   THE USE OF RADIO-BROMINATED PARA-BROMOSPIROPERIDOL FOR GAMMA-RAY IMAGING OF DOPAMINE-RECEPTORS [J].
FRIEDMAN, AM ;
HUANG, CC ;
KULMALA, HA ;
DINERSTEIN, R ;
NAVONE, J ;
BRUNSDEN, B ;
GAWLAS, D ;
COOPER, M .
INTERNATIONAL JOURNAL OF NUCLEAR MEDICINE & BIOLOGY, 1982, 9 (01) :57-&
[8]   REGIONAL STUDIES OF CATECHOLAMINES IN RAT BRAIN .I. DISPOSITION OF [3H]NOREPINEPHRINE [3H]DOPAMINE AND [3H]DOPA IN VARIOUS REGIONS OF BRAIN [J].
GLOWINSKI, J ;
IVERSEN, LL .
JOURNAL OF NEUROCHEMISTRY, 1966, 13 (08) :655-+
[9]   DEMONSTRATION OF NEUROLEPTIC RECEPTOR-SITES IN MOUSE-BRAIN BY AUTORADIOGRAPHY [J].
HOLLT, V ;
SCHUBERT, P .
BRAIN RESEARCH, 1978, 151 (01) :149-153
[10]   DEMONSTRATION INVIVO OF SPECIFIC BINDING-SITES FOR NEUROLEPTIC DRUGS IN MOUSE-BRAIN [J].
HOLLT, V ;
CZLONKOWSKI, A ;
HERZ, A .
BRAIN RESEARCH, 1977, 130 (01) :176-183