ORGAN SELECTIVITY OF HEXAHYDROSILADIFENIDOL IN BLOCKING PREJUNCTIONAL AND POSTJUNCTIONAL MUSCARINIC RECEPTORS STUDIED IN GUINEA-PIG ILEUM AND RAT-HEART

被引:57
作者
FUDER, H [1 ]
KILBINGER, H [1 ]
MULLER, H [1 ]
机构
[1] UNIV MAINZ,INST PHARMAKOL,OBERE ZAHLBACHER STR 67,D-6500 MAINZ,FED REP GER
关键词
D O I
10.1016/0014-2999(85)90352-8
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:125 / 127
页数:3
相关论文
共 9 条
[1]   COMPARISON OF AFFINITY CONSTANTS FOR MUSCARINE-SENSITIVE ACETYLCHOLINE RECEPTORS IN GUINEA-PIG ATRIAL PACEMAKER CELLS AT 29 DEGREESC AND IN ILEUM AT 29 DEGREESC AND 37 DEGREESC [J].
BARLOW, RB ;
BERRY, KJ ;
GLENTON, PAM ;
NIKOLAOU, NM ;
SOH, KS .
BRITISH JOURNAL OF PHARMACOLOGY, 1976, 58 (04) :613-620
[2]   MUSCARINIC RECEPTOR SUBCLASSES [J].
BIRDSALL, NJM ;
HULME, EC .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1983, 4 (11) :459-463
[3]   SYMPATHETIC-NERVE STIMULATION ON THE PERFUSED RAT-HEART - AFFINITIES OF N-METHYLATROPINE AND PIRENZEPINE AT PRE-SYNAPTIC AND POSTSYNAPTIC MUSCARINE RECEPTORS [J].
FUDER, H ;
RINK, D ;
MUSCHOLL, E .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1982, 318 (03) :210-219
[4]   THE EFFECTS OF SEVERAL MUSCARINIC ANTAGONISTS ON PRESYNAPTIC AND POSTSYNAPTIC RECEPTORS IN THE ISOLATED RABBIT HEART [J].
FUDER, H ;
MEISER, C ;
WORMSTALL, H ;
MUSCHOLL, E .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1981, 316 (01) :31-37
[5]   AFFINITY AND EFFICACY OF RACEMIC, (+)-METHACHOLINE, AND (-)-METHACHOLINE IN MUSCARINIC INHIBITION OF [H-3]-NORADRENALINE RELEASE [J].
FUDER, H ;
JUNG, B .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 84 (02) :477-487
[6]   COMPARISON OF AFFINITIES OF MUSCARINIC ANTAGONISTS TO PREJUNCTIONAL AND POSTJUNCTIONAL RECEPTORS IN THE GUINEA-PIG ILEUM [J].
KILBINGER, H ;
HALIM, S ;
LAMBRECHT, G ;
WEILER, W ;
WESSLER, I .
EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 103 (3-4) :313-320
[7]   2 TYPES OF NEURONAL MUSCARINE RECEPTORS MODULATING ACETYLCHOLINE-RELEASE FROM GUINEA-PIG MYENTERIC PLEXUS [J].
KILBINGER, H ;
NAFZIGER, M .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1985, 328 (03) :304-309
[8]  
LAMBRECHT G, 1984, Naunyn-Schmiedeberg's Archives of Pharmacology, V325, pR62
[9]  
MUTSCHLER E, 1984, TRENDS PHARM SCI S39, V5