BICUCULLINE-INSENSITIVE GABA RECEPTORS - STUDIES ON THE BINDING OF (-)-BACLOFEN TO RAT CEREBELLAR MEMBRANES

被引:157
作者
DREW, CA [1 ]
JOHNSTON, GAR [1 ]
WEATHERBY, RP [1 ]
机构
[1] UNIV SYDNEY,DEPT PHARMACOL,SYDNEY,NSW 2006,AUSTRALIA
关键词
D O I
10.1016/0304-3940(84)90181-2
中图分类号
Q189 [神经科学];
学科分类号
071006 ;
摘要
引用
收藏
页码:317 / 321
页数:5
相关论文
共 15 条
[1]  
ALLAN RD, 1980, J NEUROCHEM, V34, P651
[2]  
AULT B, 1983, SOC NEUR ABSTR, V9, P411
[3]   CHARACTERISTICS OF GABAB RECEPTOR-BINDING SITES ON RAT WHOLE BRAIN SYNAPTIC-MEMBRANES [J].
BOWERY, NG ;
HILL, DR ;
HUDSON, AL .
BRITISH JOURNAL OF PHARMACOLOGY, 1983, 78 (01) :191-206
[4]   BACLOFEN - 10 YEARS ON [J].
BOWERY, NG .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1982, 3 (10) :400-403
[5]   (-) BACLOFEN DECREASES NEUROTRANSMITTER RELEASE IN THE MAMMALIAN CNS BY AN ACTION AT A NOVEL GABA RECEPTOR [J].
BOWERY, NG ;
HILL, DR ;
HUDSON, AL ;
DOBLE, A ;
MIDDLEMISS, DN ;
SHAW, J ;
TURNBULL, M .
NATURE, 1980, 283 (5742) :92-94
[6]  
BURGISSER E, 1981, MOL PHARMACOL, V19, P205
[7]   CENTRAL EFFECTS OF BETA-(PARA-CHLOROPHENYL)-GAMMA-AMINOBUTYRIC ACID [J].
CURTIS, DR ;
GAME, CJA ;
JOHNSTON, GA ;
MCCULLOCH, RM .
BRAIN RESEARCH, 1974, 70 (03) :493-499
[8]   ACTION OF BETA-PHENYL-GABA DERIVATIVES ON NEURONS OF CAT CEREBRAL-CORTEX [J].
DAVIES, J ;
WATKINS, JC .
BRAIN RESEARCH, 1974, 70 (03) :501-505
[9]   BACLOFEN-H-3 AND H-3-GABA BIND TO BICUCULLINE-INSENSITIVE GABA-B SITES IN RAT-BRAIN [J].
HILL, DR ;
BOWERY, NG .
NATURE, 1981, 290 (5802) :149-152
[10]  
Johnston, 1976, GABA NERVOUS SYSTEM, P394