CYCLIC SOMATOSTATIN OCTAPEPTIDE ANALOGS WITH HIGH-AFFINITY AND SELECTIVITY TOWARD MU OPIOID RECEPTORS

被引：109

作者：

GULYA, K

PELTON, JT

HRUBY, VJ

YAMAMURA, HI

机构：

[1] UNIV ARIZONA,DEPT CHEM,TUCSON,AZ 85721

[2] UNIV ARIZONA,HLTH SCI CTR,DEPT PHARMACOL,TUCSON,AZ 85724

来源：

LIFE SCIENCES | 1986年 / 38卷 / 24期

关键词：

D O I：

10.1016/0024-3205(86)90574-6

中图分类号：

R-3 [医学研究方法]; R3 [基础医学];

学科分类号：

1001 ;

摘要：

引用

页码：2221 / 2229

页数：9

共 21 条

[1] CHARACTERIZATION OF [H-3][ 2-D-PENICILLAMINE, 5-D-PENICILLAMINE] ENKEPHALIN BINDING TO DELTA-OPIATE RECEPTORS IN THE RAT-BRAIN AND NEUROBLASTOMA-GLIOMA HYBRID CELL-LINE (NG-108-15) [J].

AKIYAMA, K ;

GEE, KW ;

MOSBERG, HI ;

HRUBY, VJ ;

YAMAMURA, HI .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1985, 82 (08) :2543-2547

[2] INTERACTION OF LIGANDS WITH OPIATE RECEPTORS OF BRAIN MEMBRANES - REGULATION BY IONS AND NUCLEOTIDES [J].

BLUME, AJ .

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1978, 75 (04) :1713-1717

[3]

BOTHMAN RB, 1985, MOL PHARM, V27, P399

[4] REGIONAL DISTRIBUTION OF SOMATOSTATIN IN RAT-BRAIN [J].

BROWNSTEIN, M ;

ARIMURA, A ;

SATO, H ;

SCHALLY, AV ;

KIZER, JS .

ENDOCRINOLOGY, 1975, 96 (06) :1456-1461

[5]

CHANG KJ, 1979, J BIOL CHEM, V254, P2610

[6]

CZERNIK A, 1983, J BIOL CHEM, V258, P2325

[7] CHARACTERIZATION, REGIONAL DISTRIBUTION, AND SUB-CELLULAR DISTRIBUTION OF I-125-TYR1-SOMATOSTATIN BINDING-SITES IN RAT-BRAIN [J].

EPELBAUM, J ;

ARANCIBIA, LT ;

KORDON, C ;

ENJALBERT, A .

JOURNAL OF NEUROCHEMISTRY, 1982, 38 (06) :1515-1523

[8] SUBCELLULAR-DISTRIBUTION OF RADIOIMMUNOASSAYABLE SOMATOSTATIN IN RAT-BRAIN [J].

EPELBAUM, J ;

BRAZEAU, P ;

TSANG, D ;

BRAWER, J ;

MARTIN, JB .

BRAIN RESEARCH, 1977, 126 (02) :309-323

[9] THE IMMUNO-CYTOCHEMICAL LOCALIZATION OF SOMATOSTATIN-CONTAINING NEURONS IN THE RAT CENTRAL NERVOUS-SYSTEM [J].

FINLEY, JCW ;

MADERDRUT, JL ;

ROGER, LJ ;

PETRUSZ, P .

NEUROSCIENCE, 1981, 6 (11) :2173-2192

[10]

GULYA K, 1985, J PHARMACOL EXP THER, V235, P254

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