INVITRO INHIBITION OF PLASMODIUM-FALCIPARUM BY PYRAZOFURIN, AN INHIBITOR OF PYRIMIDINE BIOSYNTHESIS DE NOVO

被引:45
作者
SCOTT, HV [1 ]
GERO, AM [1 ]
OSULLIVAN, WJ [1 ]
机构
[1] UNIV NEW S WALES, SCH BIOCHEM, KENSINGTON, NSW 2033, AUSTRALIA
关键词
D O I
10.1016/0166-6851(86)90045-9
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:3 / 15
页数:13
相关论文
共 30 条
[1]  
BUNGENER W, 1967, Z TROPENMED PARASIT, V18, P456
[2]  
Cleland W W, 1979, Methods Enzymol, V63, P103
[3]   QUANTITATIVE ASSESSMENT OF ANTI-MALARIAL ACTIVITY INVITRO BY A SEMIAUTOMATED MICRODILUTION TECHNIQUE [J].
DESJARDINS, RE ;
CANFIELD, CJ ;
HAYNES, JD ;
CHULAY, JD .
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 1979, 16 (06) :710-718
[4]  
DIX DE, 1979, CANCER RES, V39, P4485
[5]  
FIELD JW, 1956, MICROSCOPIC DIAGNO 2
[6]   STUDIES ON COORDINATE ACTIVITY AND LABILITY OF OROTIDYLATE PHOSPHORIBOSYLTRANSFERASE AND DECARBOXYLASE IN HUMAN ERYTHROCYTES, AND EFFECTS OF ALLOPURINOL ADMINISTRATION [J].
FOX, RM ;
WOOD, MH ;
OSULLIVA.WJ .
JOURNAL OF CLINICAL INVESTIGATION, 1971, 50 (05) :1050-&
[7]   DIHYDROOROTATE DEHYDROGENASE, OROTATE PHOSPHORIBOSYLTRANSFERASE AND OROTIDINE-5'-PHOSPHATE DECARBOXYLASE IN PLASMODIUM-FALCIPARUM [J].
GERO, AM ;
TETLEY, K ;
COOMBS, GH ;
PHILLIPS, RS .
TRANSACTIONS OF THE ROYAL SOCIETY OF TROPICAL MEDICINE AND HYGIENE, 1981, 75 (05) :719-720
[8]   PYRIMIDINE DENOVO SYNTHESIS DURING THE LIFE-CYCLE OF THE INTRAERYTHROCYTIC STAGE OF PLASMODIUM-FALCIPARUM [J].
GERO, AM ;
BROWN, GV ;
OSULLIVAN, WJ .
JOURNAL OF PARASITOLOGY, 1984, 70 (04) :536-541
[9]   SYNERGISTIC EFFECT OF PURINE DERIVATIVES ON THE TOXICITY OF PYRAZOFURIN AND 6-AZAURIDINE TOWARDS CULTURED MAMMALIAN-CELLS [J].
GUPTA, RS ;
MOFFAT, MRK .
JOURNAL OF CELLULAR PHYSIOLOGY, 1982, 111 (03) :291-294
[10]   BIOCHEMISTRY AND BIOLOGICAL EFFECTS OF PYRAZOFURINS (PYRAZOMYCINS) - INITIAL CLINICAL-TRIAL [J].
GUTOWSKI, GE ;
SWEENEY, MJ ;
DELONG, DC ;
HAMILL, RL ;
GERZON, K ;
DYKE, RW .
ANNALS OF THE NEW YORK ACADEMY OF SCIENCES, 1975, 255 (AUG8) :544-551